Dynorphin A (1-10) (TFA), an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor . Dynorphin A (1-10) (TFA) also blocks NMDA -activated current with an IC 50 of 42.0 μM.
Appearance:Solid
IC50& Target:NMDA Receptor κ Opioid Receptor/KOR
In Vitro:Dynorphin A (1-10) (TFA), an endogenous opioid neuropeptide, binds in the transmembrane domain of the κ-receptor. The non-opioid actions of various forms of Dynorphin A (DynA) are examined on N-methyl-D-aspartate (NMDA) receptor channels in isolated
Biological Activity:Dynorphin A (1-10) (TFA), an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor . Dynorphin A (1-10) (TFA) also blocks NMDA -activated current with an IC 50 of 42.0 μM.
Specifications
Specifications & Purity
≥98%
Storage
Desiccated,Store at -80°C
Shipped In
Dry ice packs + Cold packs
This product requires cold chain shipping. Ground and other economy services are not available.
Action Type
AGONIST
Purity
≥98%
Names and Identifiers
Molecular Weight
1348.48
Advanced Data
Certificates (CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Chemical and Physical Properties
Solubility
DMSO : 100 mg/mL (74.16 mM; Need ultrasonic) H2O : 50 mg/mL (37.08 mM; Need ultrasonic)
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