DFMTI - 10mM in DMSO , CAS No.864864-86-8

CAS: 864864-86-8 Cat. No.: D655144 Formule: C₂₀H₁₈F₂N₄O Poids moléculaire: 368.38

GRADE & PURITY 10mM in DMSO

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

Vue d’ensemble

DFMTI can completely block the rmGlu1 L757V glutamate response.In vitro: DFMTI can completely block the rmGlu1 L757V glutamate response, although significantly higher concentrations were required to induce blockade.In vivo: DFMTI is efficacious in disrupting prepulse inhibition when dosed orally in rats. DFMTI exhibits a moderate decrease in human potency of approximately 3-fold when compared to rat, exemplified by DFMTI.

IC50& Target:mGluR1

Specifications

Spécifications et pureté

10mM in DMSO

Mécanismes biochimiques et physiologiques

DFMTI can completely block the rmGlu1 L757V glutamate response.\nIn vitro: DFMTI can completely block the rmGlu1 L757V glutamate response, although significantly higher concentrations were required to induce blockade.\nIn vivo: DFMTI is efficacious in dis

Conditions de stockage de stockage

Store at -80°C

Expédié en

Dry ice packs + Cold packs

Ce produit nécessite l'expédition en chaîne froide. Les services terrestres et autres services économiques ne sont pas disponibles.

Type d'action

INHIBITOR

Noms et identifiants

• Poids moléculaire: 368.38