EHMT2-IN-1 , CAS No.2230849-55-3

CAS: 2230849-55-3 Cat. No.: E646651 分子式: C₁₈H₂₃N₇O 分子量: 353.42 PubChem CID: 135154879

Storage

Store at -20°C

Shipped In

Ice chest + Ice pads

概要

EHMT2-IN-1 is a potent EHMT inhibitor, with IC 50 s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer

In Vitro

EHMT2-IN-1 (Compound 108) potent EHMT inhibitor, with IC 50 s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Form:Solid

IC50& Target:EHMTI PEP <100 nM (IC 50 ) EHMT2 PEP <100 nM (IC 50 ) EHMT2 ICW <100 nM (IC 50 )

Specifications

生化学的・生理学的メカニズム

EHMT2-IN-1 is a potent EHMT inhibitor, with IC 50 s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer.

保管条件

Store at -20°C

入荷

Ice chest + Ice pads

この製品は冷冷この冷このこの製品の運送が必要です。地上およびその他の経済サービスは利用できません。

アクションタイプ

INHIBITOR

名前と識別子

• カノニカル・スマイル: CC1=CC(=NC(=N1)NC2=CC(=C(C=C2)OC)N3C=C(C=N3)CNC)NC
• IUPAC Name: 2-N-[4-methoxy-3-[4-(methylaminomethyl)pyrazol-1-yl]phenyl]-4-N,6-dimethylpyrimidine-2,4-diamine
• InChIKey: DJSJHTKOFPOYRZ-UHFFFAOYSA-N
• INCHI: 1S/C18H23N7O/c1-12-7-17(20-3)24-18(22-12)23-14-5-6-16(26-4)15(8-14)25-11-13(9-19-2)10-21-25/h5-8,10-11,19H,9H2,1-4H3,(H2,20,22,23,24)
• PubChem CID: 135154879
• 分子量: 353.42

化学的性質と物理的性質

• 溶解度: DMSO : 55 mg/mL (155.62 mM; Need ultrasonic)