EHMT2-IN-2 - ≥99% , CAS No.2230850-47-0

CAS: 2230850-47-0 Cat. No.: E648205 分子式: C₂₁H₂₂N₆O 分子量: 374.44 PubChem CID: 135154251

GRADE & PURITY ≥99%

Storage

Store at -20°C

Shipped In

Ice chest + Ice pads

概要

EHMT2-IN-2 is a potent EHMT inhibitor, with IC 50 s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disease or cancer

In Vitro

EHMT2-IN-2 (Compound 200) is a potent EHMT inhibitor, with IC 50 s of all < 100 nM for EEHMT1 peptide, EHMT2 peptide and cellular EHMT2. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Form:Solid

IC50& Target:EHMTI PEP <100 nM (IC 50 ) EHMT2 PEP <100 nM (IC 50 ) EHMT2 ICW <100 nM (IC 50 )

Specifications

仕様と純度

≥99%

生化学的・生理学的メカニズム

EHMT2-IN-2 is a potent EHMT inhibitor, with IC 50 s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disease or cancer.

保管条件

Store at -20°C

入荷

Ice chest + Ice pads

この製品は冷冷この冷このこの製品の運送が必要です。地上およびその他の経済サービスは利用できません。

アクションタイプ

INHIBITOR

純度

≥99%

名前と識別子

• カノニカル・スマイル: CC1=CC(=NC(=N1)NC2=CC(=C(C=C2)OC)C3=C(C4=C(N3)C=NC=C4)C)NC
• IUPAC Name: 2-N-[4-methoxy-3-(3-methyl-1H-pyrrolo[2,3-c]pyridin-2-yl)phenyl]-4-N,6-dimethylpyrimidine-2,4-diamine
• InChIKey: AZRYONWATLLNFX-UHFFFAOYSA-N
• INCHI: 1S/C21H22N6O/c1-12-9-19(22-3)27-21(24-12)25-14-5-6-18(28-4)16(10-14)20-13(2)15-7-8-23-11-17(15)26-20/h5-11,26H,1-4H3,(H2,22,24,25,27)
• PubChem CID: 135154251
• 分子量: 374.44

化学的性質と物理的性質

• 溶解度: DMSO : 50 mg/mL (133.53 mM; Need ultrasonic)