ERAP2-IN-1 (compound 61) is an uncompetitive ERAP2 inhibitor. ERAP2-IN-1 specifically inhibits the ERAP2 peptide hydrolysis activity, inhibiting Arg-AMC hydrolysis with an IC 50 of 27 μM and model peptide hydrolysis with an IC 50 of 44 μM.
仕様
仕様と純度
10mM in DMSO
生化学的・生理学的メカニズム
ERAP2-IN-1 (compound 61) is an uncompetitive ERAP2 inhibitor. ERAP2-IN-1 specifically inhibits the ERAP2 peptide hydrolysis activity, inhibiting Arg-AMC hydrolysis with an IC 50 of 27 μM and model peptide hydrolysis with an IC 50 of 44 μM.
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よくある質問
How should this product be stored?
Store at ?80 °C. Ultra-low temperature storage is required to maintain the specified shelf life.
How is this product shipped?
This product ships frozen with dry ice and cold packs. Unpack on arrival and transfer it to the storage condition stated above; handle dry ice with insulated gloves in a ventilated area.
What are the CAS number, molecular formula and molecular weight?
The CAS Number is 2420551-38-6, the molecular formula is C20H21F3N2O5S, and the molecular weight is 458.45 g/mol.
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