S961 TFA , CAS No.S659083

CAS: S659083 Cat. No.: S659083 分子式: C₂₁₁H₂₉₇N₅₅O₇₁S₂.C₂HF₃O₂ 分子量: 4918.15

Storage

Protected from light,Desiccated,Store at -80°C

Shipped In

Dry ice packs + Cold packs

概要

S961 TFA is an high-affinity and selective insulin receptor ( IR ) antagonist with IC 50 s of 0.048, 0.027, and 630 nM for HIR-A, HIR-B, and human insulin-like growth factor I receptor (HIGF-IR) in SPA-assay, respectively.

Appearance:Solid

In Vitro:S961 also shows high-affinity to Rat IR and Pig IR with IC 50 s of 0.056 nM and 0.084 nM in PEG-assay, respectively. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Biological Activity:S961 TFA is an high-affinity and selective insulin receptor ( IR ) antagonist with IC 50 s of 0.048, 0.027, and 630 nM for HIR-A, HIR-B, and human insulin-like growth factor I receptor (HIGF-IR) in SPA-assay, respectively.

仕様

保管条件

Protected from light,Desiccated,Store at -80°C

入荷

Dry ice packs + Cold packs

この製品は冷冷この冷このこの製品の運送が必要です。地上およびその他の経済サービスは利用できません。

名前と識別子

分子量

4918.15

化学的性質と物理的性質

• 溶解度: H2O : 6.5 mg/mL (1.32 mM; ultrasonic and adjust pH to 12 with NaOH)