UCSF924 - 10mM in DMSO , CAS No.1434515-70-4

CAS: 1434515-70-4 Cat. No.: U655068 分子式: C₂₀H₂₂N₂O₂ 分子量: 322.40

GRADE & PURITY 10mM in DMSO

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

概要

UCSF924 is a potent and specific dopamine D4 receptor (DRD4) partial agonist with a EC 50 of 4.2 nM. UCSF924 has a high-affinity with a K i value of 3 nM for DRD4 and shows no measurable affinity for D2, D3 or the F261V/L328F D4 mutant. UCSF924 is a 7.4-fold bias toward arrestin over Gαi/o signaling, referenced to quinpirole

IC50& Target:Ki: 3 nM (dopamine D4 receptor)

Specifications

仕様と純度

10mM in DMSO

生化学的・生理学的メカニズム

UCSF924 is a potent and specific dopamine D4 receptor (DRD4) partial agonist with a EC 50 of 4.2 nM. UCSF924 has a high-affinity with a K i value of 3 nM for DRD4 and shows no measurable affinity for D2, D3 or the F261V/L328F D4 mutant. UCSF924 is a 7.4-f

保管条件

Store at -80°C

入荷

Dry ice packs + Cold packs

この製品は冷冷この冷このこの製品の運送が必要です。地上およびその他の経済サービスは利用できません。

名前と識別子

• 分子量: 322.40

よくある質問

How should this product be stored?

Store at ?80 °C. Ultra-low temperature storage is required to maintain the specified shelf life.

How is this product shipped?

This product ships frozen with dry ice and cold packs. Unpack on arrival and transfer it to the storage condition stated above; handle dry ice with insulated gloves in a ventilated area.

What are the CAS number, molecular formula and molecular weight?

The CAS Number is 1434515-70-4, the molecular formula is C20H22N2O2, and the molecular weight is 322.40 g/mol.

What documentation is provided?

Available product documentation, including Certificates of Analysis (COA), Safety Data Sheets (SDS), and specification sheets, is shown in the product document area. Document availability and access follow the current site policy.