BCX 1470 methanesulfonate - Moligand™,≥99% , CAS No.217099-44-0

CAS: 217099-44-0 Cat. No.: B647162 Molecular Weight: 398.48
AVAILABLE TO ORDER
GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥99%
Synonyms
2-Thiophenecarboxylic acid 2-(aminoiminomethyl)benzo[b]thiophen-6-yl ester methanesulfonate | 2-Carbamimidoylbenzo[b]thiophen-6-yl thiophene-2-carboxylate methanesulfonate
Storage
Protected from light,Store at -20°C,Argon charged,Desiccated
Shipped In
Ice chest + Ice pads
 ·  off list, applied to all prices below.
Size
Status
Price
Qty
5mg
B647162-5mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$68.90
1mg
B647162-1mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$19.90
25mg
B647162-25mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$239.90
100mg
B647162-100mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$689.90
Enter a quantity for the sizes you want to add.
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Why this grade

Moligand™,≥99% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

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Storage & shipping

Protected from light,Store at -20°C,Argon charged,Desiccated Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.

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Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

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Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Overview

BCX 1470 methanesulfonate inhibits the esterolytic activity of factor D ( IC 50 =96 nM) and C1s ( IC 50 =1.6 nM), 3.4- and 200-fold better, respectively, than that of trypsin.

In Vitro

BCX 1470 methanesulfonate is serine protease inhibitor. BCX 1470 methanesulfonate blocks the esterolytic and hemolytic activities of the complement enzymes Cls and factor D in vitro, also blocked development of RPA-induced edema in the rat. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Form:Solid

IC50& Target:IC50: 96 nM (Factor D),1.6 nM (C1s),326 nM (Trypsin)

Specifications

Synonyms
2-Thiophenecarboxylic acid 2-(aminoiminomethyl)benzo[b]thiophen-6-yl ester methanesulfonate | 2-Carbamimidoylbenzo[b]thiophen-6-yl thiophene-2-carboxylate methanesulfonate
Specifications & Purity
Moligand™, ≥99%
Biochemical and Physiological Mechanisms
BCX 1470 methanesulfonate inhibits the esterolytic activity of factor D ( IC 50 =96 nM) and C1s ( IC 50 =1.6 nM), 3.4- and 200-fold better, respectively, than that of trypsin.
Storage
Protected from light, Store at -20°C, Argon charged, Desiccated
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Grade
Moligand™
Action Type
INHIBITOR
Purity
≥99%
Names and Identifiers
Alternate CAS 217099-43-9
Molecular Weight 398.48

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Certificates(CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Chemical and Physical Properties
SolubilityDMSO : ≥ 33.33 mg/mL (83.64 mM)
SensitivityMoisture sensitive
Solution Calculators
Reviews

Customer Reviews

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