BQ-3020 TFA salt - Moligand™, ≥98% , Agonist of ET B receptor, CAS No.143113-45-5（free basis）, Agonist of ET B receptor

CAS: 143113-45-5（free basis） Cat. No.: B287102 Formula: C₉₆H₁₄₀N₂₀O₂₅S（free basis） Peso molecolare: 2006.32（free basis） Numero EC: 686-390-9

GRADE & PURITY Moligand™, ≥98%

Synonyms

Acetyl-(Ala 11,15)-ET 1 (6-21) TFA salt | Acetyl-[Ala 11,15]-endothelin 1 (6-21) TFA salt

Storage

Protected from light,Store at -20°C,Desiccated

Shipped In

Ice chest + Ice pads

Specifications

Sinonimi

Acetyl-(Ala 11,15)-ET 1 (6-21) TFA salt | Acetyl-[Ala 11,15]-endothelin 1 (6-21) TFA salt

Specifiche e purezza

Moligand™, ≥98%

Meccanismi biochimici e fisiologici

Highly potent and selective ETBendothelin receptor agonist (Kivalues are 0.18 and 970 nM at human ETBand ETAreceptors respectively).

Condizioni di conservazione di stoccaggio

Protected from light,Store at -20°C,Desiccated

Spedito in

Ice chest + Ice pads

Questo prodotto richiede spedizione a catena fredda. I servizi di terra e altri servizi economici non sono disponibili.

Grado

Moligand™

Tipo di azione

AGONIST

Meccanismo d'azione

Agonist of ET B receptor

Purezza

≥98%

Nomi e identificatori

Sorrisi canonici

CC[C@H](C)[C@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC1=CNC=N1)NC(=O)[C@H](C)NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)[C@H](CC1=CC=C(O)C=C1)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCSC)NC(=O)[

InChIKey

AYJUXFCWNAVJLN-FHOIYVHLSA-N

Isomeri SMILES

CC[C@H](C)[C@@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC1=CNC2=CC=CC=C21)C(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC3=CN=CN3)NC(=O)[C@H](C)NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@H](CC5=CC=C(C=C5)O)NC(=O)[C@H](C(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](CC(C)C)NC(=O)C

Peso molecolare

2006.32（free basis）

Reaxy-Rn

24249740

Reaxys-RN_link_address

https://www.reaxys.com/reaxys/secured/hopinto.do?context=S&query=IDE.XRN=24249740&ln=

Obiettivi associati (umani)

EDNRB Tclin Endothelin receptor type B (0 Activities)

Discover Target: EDNRB

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Proprietà chimiche e fisiche

• Solubilità: Soluble to 0.50 (mg/mL) in sodium bicarbonate (0.03M)
• Sensibilità: Light sensitive