Casopitant mesylate - Moligand™, 10 mM in DMSO , CAS No.414910-30-8

CAS: 414910-30-8 Cat. No.: C1497018 Formula: C₃₁H₃₉F₇N₄O₅S Peso molecolare: 712.72 Numero EC: 638-762-7 PubChem CID: 11686295

GRADE & PURITY Moligand™, 10 mM in DMSO

Storage

Desiccated,Store at -80°C

Shipped In

Dry ice packs + Cold packs

Panoramica

Casopitant mesylate (GW679769B) is a potent, selective, brain permeable and orally active neurokinin 1 ( NK1 ) receptor antagonist. Casopitant mesylate is a second in the class of antiemetics that acts to antagonise the emetogenic effect of Substance P. Casopitant mesylate is also a substrate and a weak-to-moderate inhibitor of CYP3A4 . Casopitant mesylate can be used for chemotherapy-induced nausea and vomiting (CINV) and postoperative nausea and vomiting (PONV) .

Specifications

Specifiche e purezza

Moligand™, 10 mM in DMSO

Condizioni di conservazione di stoccaggio

Desiccated,Store at -80°C

Spedito in

Dry ice packs + Cold packs

Questo prodotto richiede spedizione a catena fredda. I servizi di terra e altri servizi economici non sono disponibili.

Grado

Moligand™

Tipo di azione

ANTAGONIST

Nomi e identificatori

• Isomeri SMILES: CC1=C(C=CC(=C1)F)[C@H]2C[C@H](CCN2C(=O)N(C)[C@H](C)C3=CC(=CC(=C3)C(F)(F)F)C(F)(F)F)N4CCN(CC4)C(=O)C.CS(=O)(=O)O
• PubChem CID: 11686295
• Peso molecolare: 712.72