CBP/p300-IN-10 - ≥98% , CAS No.2259641-71-7

CAS: 2259641-71-7 Cat. No.: C648970 Formula: C₂₅H₂₄F₅N₅O₃ Peso molecolare: 537.48

GRADE & PURITY ≥98%

Storage

Store at -20°C

Shipped In

Ice chest + Ice pads

Panoramica

CBP/p300-IN-10 is a highly potent histone acetyltransferase EP300 and CREBBP with IC 50 values of 26 nM and 39 nM, respectively. CBP/p300-IN-10 can be used to research anticancer

In Vitro

CBP/p300-IN-10 (example 84) (0-1 μM; 3 h) inhibit H3K27Ac activity in LK2 cells with an IC 50 of 22 nM. CBP/p300-IN-10 (38 nM-10 mM; 3 days) has inhibitory activity against LK2 and TE-8. MCE has not independently confirmed the accuracy of these methods. They are for reference only. Cell Proliferation AssayCell Line: LK2 and TE-8 Concentration: 38 nM-10 mM Incubation Time: 3 days Result: Inhibited LK2 and TE-8 with GI 50 s of 97.163 nM and 152.484 nM, respectively.

Form:Solid

IC50& Target:EP300 26 nM (IC 50 ) CREBBP 39 nM (IC 50 )

Specifications

Specifiche e purezza

≥98%

Meccanismi biochimici e fisiologici

CBP/p300-IN-10 is a highly potent histone acetyltransferase EP300 and CREBBP with IC 50 values of 26 nM and 39 nM, respectively. CBP/p300-IN-10 can be used to research anticancer.

Condizioni di conservazione di stoccaggio

Store at -20°C

Spedito in

Ice chest + Ice pads

Questo prodotto richiede spedizione a catena fredda. I servizi di terra e altri servizi economici non sono disponibili.

Tipo di azione

INHIBITOR

Purezza

≥98%

Nomi e identificatori

Peso molecolare

537.48

Proprietà chimiche e fisiche

• Solubilità: DMSO : 10.5 mg/mL (19.54 mM; ultrasonic and warming and heat to 80°C)