FSHR agonist 1 - ≥98% , CAS No.1256776-89-2

CAS: 1256776-89-2 Cat. No.: F646397 Molecular Weight: 467.62
AVAILABLE TO ORDER
GRADE & PURITY ≥98%
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
 ·  off list, applied to all prices below.
Size
Status
Price
Qty
1mg
F646397-1mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$560.90
5mg
F646397-5mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$1,700.90
10mg
F646397-10mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
$2,700.90
Enter a quantity for the sizes you want to add.
🧪

Why this grade

≥98% for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

🌡

Storage & shipping

Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.

📋

Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

📚

Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Overview

FSHR agonist 1 is a high affinity and allosteric follicle stimulating hormone receptor (FSHR) agonist with a pEC 50 of 7.72. FSHR agonist 1 formes extensive interactions with the TMD to directly activate FSHR

In Vitro

The binding of FSHR agonist 1 (compound 21f) to the FSHR TMD pocket induces inward movements of TM6 and TM7, which directly results in FSHR activation. FSHR agonist 1 (compound 21f) can activate FSHR, LHCGR and TSHR with highly potency and efficacy, while the activation potency for FSHR is more than 10-fold higher than LHCGR (pEC 50 of 6.26) and TSHR (pEC 50 of 6.48). MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Form:Solid

IC50& Target:pEC50: 7.72 (FSHR)

Specifications

Specifications & Purity
≥98%
Biochemical and Physiological Mechanisms
FSHR agonist 1 is a high affinity and allosteric follicle stimulating hormone receptor (FSHR) agonist with a pEC 50 of 7.72. FSHR agonist 1 formes extensive interactions with the TMD to directly activate FSHR.
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
This product requires cold chain shipping. Ground and other economy services are not available.
Action Type
AGONIST
Purity
≥98%
Names and Identifiers
Molecular Weight 467.62

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Certificates(CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Chemical and Physical Properties
SolubilityDMSO : 50 mg/mL (106.92 mM; Need ultrasonic)
Solution Calculators
Reviews

Customer Reviews

Shall we send you a message when we have discounts available?

Remind me later

Thank you! Please check your email inbox to confirm.

Oops! Notifications are disabled.