Gallamine Triethiodide - Moligand™, 10mM in DMSO , Muscle-type nicotinic acetylcholine receptor antagonist, CAS No.65-29-2, Muscle-type nicotinic acetylcholine receptor antagonist

CAS: 65-29-2 Cat. No.: G408368 Formula: C₃₀H₆₀I₃N₃O₃ Peso molecolare: 891.53 Numero EC: 200-605-1 PubChem CID: 6172

GRADE & PURITY Moligand™, 10mM in DMSO

Synonyms

2,​2',​2''-​[1,​2,​3-​benzenetriyltris(oxy​)​]​tris[N,​N,​N-​triethyl-ethanaminium, iodide (1:3)

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

Panoramica

Information

Gallamine Triethiodide Gallamine Triethiodide is a cholinergic receptor blocker with an IC50 of 68.0 ± 8.4 μM.
In vitro

In vivo

Cell Data

cell lines：

Concentrations：

Incubation Time：

Powder Purity:≥97%

Specifications

Sinonimi

2,​2',​2''-​[1,​2,​3-​benzenetriyltris(oxy​)​]​tris[N,​N,​N-​triethyl-ethanaminium, iodide (1:3)

Specifiche e purezza

Moligand™, 10mM in DMSO

Meccanismi biochimici e fisiologici

Gallamine Triethiodide is a cholinergic receptor blocker with an IC50 of 68.0 ± 8.4 μM.

Condizioni di conservazione di stoccaggio

Store at -80°C

Spedito in

Dry ice packs + Cold packs

Questo prodotto richiede spedizione a catena fredda. I servizi di terra e altri servizi economici non sono disponibili.

Grado

Moligand™

Tipo di azione

ALLOSTERIC MODULATOR, ANTAGONIST, CHANNEL BLOCKER

Meccanismo d'azione

Muscle-type nicotinic acetylcholine receptor antagonist

Nomi e identificatori

• Isomeri SMILES: CC[N+](CC)(CC)CCOC1=C(C(=CC=C1)OCC[N+](CC)(CC)CC)OCC[N+](CC)(CC)CC.[I-].[I-].[I-]
• WGK Germania: 3
• RTECS: BS1100000
• PubChem CID: 6172
• Peso molecolare: 891.53

Obiettivi associati (umani)

CHRNA1 Tclin Acetylcholine receptor subunit alpha (1 Activities)

Discover Target: CHRNA1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

CHRM2 Tclin Muscarinic acetylcholine receptor M2 (1 Activities)

Discover Target: CHRM2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Proprietà chimiche e fisiche

• Punto di fusione (°C): 235 °C

Riferimenti

1. Lin Huang, Weixia Zhang, Difei Tong, Lingzheng Lu, Weishang Zhou, Dandan Tian, Guangxu Liu, Wei Shi.  (2023)  Triclosan and triclocarban weaken the olfactory capacity of goldfish by constraining odorant recognition, disrupting olfactory signal transduction, and disturbing olfactory information processing.  WATER RESEARCH,      [PMID:36801581] [10.1016/j.watres.2023.119736]

2. Petrus Siregar, Gilbert Audira, Ling-Yi Feng, Jia-Hau Lee, Fiorency Santoso, Wen-Hao Yu, Yu-Heng Lai, Jih-Heng Li, Ying-Ting Lin, Jung-Ren Chen, Chung-Der Hsiao.  (2021)  Pharmaceutical Assessment Suggests Locomotion Hyperactivity in Zebrafish Triggered by Arecoline Might Be Associated with Multiple Muscarinic Acetylcholine Receptors Activation.  Toxins,  13  (4): (259).  [PMID:33916832] [10.3390/toxins13040259]

Domande frequenti

What is Moligand??

Moligand? is one of Aladdin Scientific's premium product lines, formulated for high-purity applications across multiple workflows. Compared to standard grades in the same workflow, Moligand? products typically offer tighter specifications, more rigorous QC, and stronger lot-to-lot consistency.

How should this product be stored?

Store at ?80 °C. Ultra-low temperature storage is required to maintain the specified shelf life.

How is this product shipped?

This product ships frozen with dry ice and cold packs. Unpack on arrival and transfer it to the storage condition stated above; handle dry ice with insulated gloves in a ventilated area.

What are the CAS number, molecular formula and molecular weight?

The CAS Number is 65-29-2, the molecular formula is C30H60I3N3O3, and the molecular weight is 891.53 g/mol.

What documentation is provided?

Available product documentation, including Certificates of Analysis (COA), Safety Data Sheets (SDS), and specification sheets, is shown in the product document area. Document availability and access follow the current site policy.