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Moligand™, ≥98% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
Cited in 21 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Product Description
Imiquimod (R 837) is an immune response modifier that acts as a toll-like receptor 7 agonist.
A TLR7 activator and angiogenesis inhibitor.
Product Application
Imiquimod is a caspase 3 activator which acts as an immunomodulator and displays antiviral and anti-tumor activity. It is a patient-applied cream used for the treatment of genital warts and basal cell carcinoma. It is also used to cure actinic keratosis on the face and scalp. It belongs to a group of drugs called immune response modifiers, which work by activating the immune system to fight abnormal skin growth.
Comprehensive hazard, handling, storage, and regulatory compliance document.
Download SDS →Lot-specific quality data. Enter your lot number to retrieve the exact COA.
Look up COA →Full quality attributes and acceptance criteria for this grade.
View spec sheet →Taxonomy Tree
| Kingdom | Organic compounds |
|---|---|
| Superclass | Organoheterocyclic compounds |
| Classe | Quinolines and derivatives |
| Subclass | Imidazoquinolines |
| Intermediate Tree Nodes | Not available |
| Direct Parent | Imidazoquinolines |
| Alternative Parents | Aminoquinolines and derivatives Imidazo-[4,5-c]pyridines Aminopyridines and derivatives N-substituted imidazoles Imidolactams Benzenoids Heteroaromatic compounds Azacyclic compounds Primary amines Organopnictogen compounds Hydrocarbon derivatives |
| Molecular Framework | Aromatic heteropolycyclic compounds |
| Substituents | Imidazoquinoline - Aminoquinoline - Imidazopyridine - Imidazo-[4,5-c]pyridine - Aminopyridine - N-substituted imidazole - Pyridine - Imidolactam - Benzenoid - Azole - Imidazole - Heteroaromatic compound - Azacycle - Organopnictogen compound - Hydrocarbon derivative - Organic nitrogen compound - Amine - Organonitrogen compound - Primary amine - Aromatic heteropolycyclic compound |
| Descrição | This compound belongs to the class of organic compounds known as imidazoquinolines. These are aromatic heterocyclic compounds containing an imidazole ring fused to a quinoline ring system. In some configurations, the imidazole ring shares a nitrogen atom with the quinoline moiety. |
| External Descriptors | imidazoquinoline |
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Find and download the COA for your product by matching the lot number on the packaging.
| Lot Number | Certificate Type | Data | Item |
|---|---|---|---|
| Certificate of Analysis | Aug 03, 2026 | I129798 | |
| Certificate of Analysis | Aug 03, 2026 | I129798 | |
| Certificate of Analysis | Aug 03, 2026 | I129798 | |
| Certificate of Analysis | Aug 03, 2026 | I129798 | |
| Certificate of Analysis | Aug 03, 2026 | I129798 | |
| Certificate of Analysis | Apr 15, 2026 | I129798 | |
| Certificate of Analysis | Nov 18, 2025 | I129798 | |
| Certificate of Analysis | Nov 18, 2025 | I129798 | |
| Certificate of Analysis | Nov 18, 2025 | I129798 | |
| Certificate of Analysis | Nov 18, 2025 | I129798 | |
| Certificate of Analysis | Nov 18, 2025 | I129798 | |
| Certificate of Analysis | Nov 18, 2025 | I129798 | |
| Certificate of Analysis | Nov 18, 2025 | I129798 | |
| Certificate of Analysis | Sep 17, 2025 | I129798 | |
| Certificate of Analysis | Aug 15, 2025 | I129798 | |
| Certificate of Analysis | Jul 30, 2025 | I129798 | |
| Certificate of Analysis | Jul 09, 2025 | I129798 | |
| Certificate of Analysis | Apr 27, 2025 | I129798 | |
| Certificate of Analysis | Nov 07, 2024 | I129798 | |
| Certificate of Analysis | Mar 12, 2024 | I129798 | |
| Certificate of Analysis | Mar 12, 2024 | I129798 | |
| Certificate of Analysis | Mar 12, 2024 | I129798 | |
| Certificate of Analysis | Mar 12, 2024 | I129798 | |
| Certificate of Analysis | Mar 12, 2024 | I129798 | |
| Certificate of Analysis | Mar 12, 2024 | I129798 | |
| Certificate of Analysis | Jan 04, 2024 | I129798 | |
| Certificate of Analysis | Apr 14, 2023 | I129798 | |
| Certificate of Analysis | Jan 03, 2023 | I129798 | |
| Certificate of Analysis | Oct 15, 2022 | I129798 | |
| Certificate of Analysis | Dec 25, 2021 | I129798 |
| Solubilidade | Soluble in DMSO (4 mg/ml ,warming to 60 °C for 15 minutes) DMF (1.5 mg/ml) at 37 °C, and water (slightly soluble) at 37 °C. Insoluble in ethanol. |
|---|---|
| Ponto de fusão (°C) | 297~299℃ |
| Peso molecular | 240.300 g/mol |
| XLogP3 | 2.600 |
| Hydrogen Bond Donor Count | 1 |
| Hydrogen Bond Acceptor Count | 3 |
| Rotatable Bond Count | 2 |
| Exact Mass | 240.137 Da |
| Monoisotopic Mass | 240.137 Da |
| Topological Polar Surface Area | 56.700 Ų |
| Heavy Atom Count | 18 |
| Formal Charge | 0 |
| Complexity | 294.000 |
| Isotope Atom Count | 0 |
| Defined Atom Stereocenter Count | 0 |
| Undefined Atom Stereocenter Count | 0 |
| Defined Bond Stereocenter Count | 0 |
| Undefined Bond Stereocenter Count | 0 |
| The total count of all stereochemical bonds | 0 |
| Covalently-Bonded Unit Count | 1 |
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