Metabolically stable inhibitor of anandamide cellular uptake (Ki= 3μM). Displays relatively low affinity for CB1and CB2receptors (Kivalues are 5.1 and > 10μM) and for vanilloid VR1 receptors (EC50= 10μM). FABP inhibitor. Has minimal activity against FAAH
Condições de armazenamento de armazenamento
Store at 2-8°C
Enviado em
Wet ice
Este produto requer transporte de cadeia fria. Serviços terrestres e outros serviços econômicos não estão disponíveis.
This compound belongs to the class of organic compounds known as amphetamines and derivatives. These are organic compounds containing or derived from 1-phenylpropan-2-amine.
External Descriptors
Not available
1. Djoumbou Feunang Y, Eisner R, Knox C, Chepelev L, Hastings J, Owen G, Fahy E, Steinbeck C, Subramanian S, Bolton E, Greiner R, and Wishart DS. ClassyFire: Automated Chemical Classification With A Comprehensive, Computable Taxonomy. Journal of Cheminformatics, 2016, 8:61.
Solvent:ethanol, Max Conc. mg/mL: 4.32, Max Conc. mM: 10; Solvent:DMSO, Max Conc. mg/mL: 4.32, Max Conc. mM: 10
Peso molecular
431.700 g/mol
XLogP3
8.000
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
3
Rotatable Bond Count
19
Exact Mass
431.34 Da
Monoisotopic Mass
431.34 Da
Topological Polar Surface Area
69.600 Ų
Heavy Atom Count
31
Formal Charge
0
Complexity
444.000
Isotope Atom Count
0
Defined Atom Stereocenter Count
1
Undefined Atom Stereocenter Count
0
Defined Bond Stereocenter Count
1
Undefined Bond Stereocenter Count
0
The total count of all stereochemical bonds
1
Covalently-Bonded Unit Count
1
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Revisões
Avaliações dos Clientes
Perguntas frequentes
What is the purity of this product?
This product is supplied at ≥98% purity (chemical assay). Lot-specific values are stated on the Certificate of Analysis.
How should this product be stored?
Store at 2–8 °C. Refrigerated storage is required to maintain the specified shelf life.
How is this product shipped?
This product ships chilled on wet ice. Unpack on arrival and transfer it to the storage condition stated above.
What are the CAS number, molecular formula and molecular weight?
The CAS Number is 616884-63-0, the molecular formula is C27H45NO3, and the molecular weight is 431.66 g/mol. InChIKey ICDMLAQPOAVWNH-HAAQQRBASA-N.
What documentation is provided?
Available product documentation, including Certificates of Analysis (COA), Safety Data Sheets (SDS), and specification sheets, is shown in the product document area. Document availability and access follow the current site policy.
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G2301434