WDR5-0102 - Moligand™,≥97% , CAS No.824960-50-1

CAS: 824960-50-1 Cat. No.: W646766 Formula: C18H19ClN4O3 Molecular Weight: 374.82
AVAILABLE TO ORDER
GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥97%
Storage
Store at 2-8°C,Protected from light
Shipped In
Wet ice
Size
USA
Germany (EU)*
Price
Qty
10mg
W646766-10mg
Made to order · 8–12 wks
$199.90
50mg
W646766-50mg
Made to order · 8–12 wks
$399.90
250mg
W646766-250mg
Made to order · 8–12 wks
$999.90
1g
W646766-1g
Made to order · 8–12 wks
$1,999.90
Enter a quantity for the sizes you want to add.
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Why this grade

Moligand™,≥97% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

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Storage & shipping

Store at 2-8°C,Protected from light Ships Wet ice Check lot-specific COA for exact specifications.

📋

Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

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Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Overview

WDR5-0102 is an inhibitor targeting WDR5-MLL1 interface (K dis =7 μM, K d =4 μM). WDR5-0102 suppresses MLL1 HMT activity, but not human H3K4 methyltransferase SETD7 and six other HMTs: G9a, EHMT1, SUV39H2, SETD8, PRMT3 , and PRMT5.

Form:Solid

Specifications

Specifications & Purity
Moligand™,≥97%
Biochemical and Physiological Mechanisms
WDR5-0102 is an inhibitor targeting WDR5-MLL1 interface (K dis =7 μM, K d =4 μM). WDR5-0102 suppresses MLL1 HMT activity, but not human H3K4 methyltransferase SETD7 and six other HMTs: G9a, EHMT1, SUV39H2, SETD8, PRMT3 , and PRMT5.
Storage
Store at 2-8°C,Protected from light
Shipped In
Wet ice
This product requires cold chain shipping. Ground and other economy services are not available.
Grade
Moligand™
Action Type
INHIBITOR
Purity
≥97%
Names and Identifiers
Molecular Weight 374.82

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Certificates(CoA,COO,BSE/TSE and Analysis Chart)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:

Find and download the COA for your product by matching the lot number on the packaging.

4 results found

Lot NumberCertificate TypeDateItem
I2603806Certificate of AnalysisMar 27, 2026 W646766
I2603815Certificate of AnalysisMar 27, 2026 W646766
I2603842Certificate of AnalysisMar 27, 2026 W646766
I2603843Certificate of AnalysisMar 27, 2026 W646766
Chemical and Physical Properties
SolubilityDMSO : 50 mg/mL (133.40 mM; ultrasonic and warming and heat to 60°C)
Solution Calculators
Reviews

Customer Reviews

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