BIBO3304 - Moligand™, 10 mM in DMSO , CAS No.191868-14-1

CAS: 191868-14-1 Cat. No.: B1494012 Molecular Weight: 529.6311402 PubChem CID: 5311021

GRADE & PURITY Moligand™, 10 mM in DMSO

Storage

Desiccated,Store at -80°C

Shipped In

Dry ice packs + Cold packs

Overview

BIBO3304 is a potent, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist, with subnanomolar affinity for both the human and the rat Y1 receptor ( IC 50 =0.38 and 0.72 nM, respectively).

Specifications

Specifications & Purity

Moligand™, 10 mM in DMSO

Storage

Desiccated, Store at -80°C

Shipped In

Dry ice packs + Cold packs

This product requires cold chain shipping. Ground and other economy services are not available.

Grade

Moligand™

Action Type

ANTAGONIST

Product Properties

• Ki Data: NPY1-R: Ki= 0.25 nM (human)

Names and Identifiers

• Isomeric SMILES: C1=CC=C(C=C1)C(C2=CC=CC=C2)C(=O)N[C@H](CCCN=C(N)N)C(=O)NCC3=CC=C(C=C3)CNC(=O)N.C(=O)(C(F)(F)F)O
• RTECS: CY1482730
• PubChem CID: 5311021
• Molecular Weight: 529.6311402

Chemical and Physical Properties

• Refractive Index: n20D~1.64 (Predicted)
• Specific Rotation[α]: α20/D -4.4°, c = 1 in DMSO