(+)-Penbutolol - 10mM in DMSO , CAS No.38363-41-6

CAS: 38363-41-6 Cat. No.: P656706 Fórmula: C₁₈H₂₉NO₂ Peso molecular: 291.43 PubChem CID: 162302

GRADE & PURITY 10mM in DMSO

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

Descripción general

(+)-Penbutolol is a β-adrenoceptor antagonist, with an IC 50 of 0.74 μM (+)-Penbutolol is an optical isomer of l-penbutolol with Na + channel-blocking action .

In Vitro

(+)-penbutolol on the [Ca 2+ ] i -increase induced by LPC is concentration-dependent. (+)-penbutolol inhibits the rounding of cells dose dependently (8±4%, 56±4% and 66±2% at the concentrations of 10 -6 M, 5×10 -6 M and 10 -5 M, respectively). MCE has not independently confirmed the accuracy of these methods. They are for reference only.

IC50& Target:IC50: 0.74 μM (β-adrenoceptor)

Specifications

Especificaciones y pureza

10mM in DMSO

Mecanismos bioquímicos y fisiológicos

(+)-Penbutolol is a β-adrenoceptor antagonist, with an IC 50 of 0.74 μM. (+)-Penbutolol is an optical isomer of l-penbutolol with Na + channel-blocking action.

Condiciones de almacenamiento de almacenamiento

Store at -80°C

Enviado en

Dry ice packs + Cold packs

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Tipo de acción

ANTAGONIST

Nombres e identificadores

• Isómeros SMILES: CC(C)(C)NC[C@H](COC1=CC=CC=C1C2CCCC2)O
• CAS alternativo: 38363-41-6
• PubChem CID: 162302
• Peso molecular: 291.43