Esplora le piccole molecole associate alla segnalazione dei GPCR e delle proteine G per lo studio della biologia dei recettori, l'analisi dei percorsi di segnalazione e lo sviluppo di test. Utilizza questa pagina per confrontare i modulatori che consentono di studiare la segnalazione a monte, i secondi messaggeri e le risposte indotte dai recettori.
GPCR/Proteina G
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9,689 prodotti
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Prodotti popolari
- Phos-tag Acrylamide AAL-107CAS: 871839-54-2 Formula: C33H38N8O3 Peso molecolare: 594.71Solido Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%◐ .Su ordinazione · 8–12 settimane Oggetto #: P1448021Visualizza prodottoPrezzi e dimensioni del pacchetto
Identificatori tecnici
- Sinonimi
- 6-(((3-(bis(pyridin-2-ylmethyl)amino)-2-hydroxypropyl)(pyridin-2-ylmethyl)amino)methyl)-N-(2-((1-hydroxyallylidene)am...
- BQ-123, Antagonist of ET A receptorCAS: 136553-81-6 Formula: C31H42N6O7 Peso molecolare: 610.7Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%● In magazzino — Magazzino negli USA, spedizione nell'EU* Oggetto #: B275090Visualizza prodottoPrezzi e dimensioni del pacchetto
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- Nome IUPAC
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- SMILES
- CC(C)CC1C(=O)NC(C(=O)NC(C(=O)N2CCCC2C(=O)NC(C(=O)N1)C(C)C)CC(=O)O)CC3=CNC4=CC=CC=C43
- InChIKey
- VYCMAAOURFJIHD-PJNXIOHISA-N
- InChI
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- Sinonimi
- 2-((3R,6S,9R,12R,17aS)-9-((1H-indol-3-yl)methyl)-6-isobutyl-3-isopropyl-1,4,7,10,13-pentaoxohexadecahydro-1H-pyrrolo[...
- GW 627368, Antagonist of EP 4 receptorCAS: 439288-66-1 Formula: C30H28N2O6S Peso molecolare: 544.62Solido Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%(HPLC)● In magazzino — Magazzino negli USA, spedizione nell'EU* Oggetto #: G288949Visualizza prodottoPrezzi e dimensioni del pacchetto
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- Nome IUPAC
- N-(benzenesulfonyl)-2-[4-(4,9-diethoxy-3-oxo-1H-benzo[f]isoindol-2-yl)phenyl]acetamide
- SMILES
- CCOC1=C2CN(C(=O)C2=C(C3=CC=CC=C31)OCC)C4=CC=C(C=C4)CC(=O)NS(=O)(=O)C5=CC=CC=C5
- InChIKey
- XREWXJVMYAXCJV-UHFFFAOYSA-N
- InChI
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- Sinonimi
- A842355 | NSC 96380 | GW627368X | GW-627368X | BCP15277 | EX-A603 | GW 627368 | SY029966 | Benzeneacetamide, 4-(4,9-d...
- PF 05190457, Antagonist of ghrelin receptorMoligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%(HPLC)● In magazzino — Magazzino negli USA, spedizione nell'EU* Oggetto #: P288410Visualizza prodottoPrezzi e dimensioni del pacchetto
Identificatori tecnici
- Nome IUPAC
- 2-(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)-1-[2-[(1R)-5-(6-methylpyrimidin-4-yl)-2,3-dihydro-1H-inden-1-yl]-2,7-diazaspiro[3.5]nonan-7-yl]ethanone
- SMILES
- CC1=CC(=NC=N1)C2=CC3=C(C=C2)C(CC3)N4CC5(C4)CCN(CC5)C(=O)CC6=CN7C=C(SC7=N6)C
- InChIKey
- ZIUDADZJCKGWKR-AREMUKBSSA-N
- InChI
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- Sinonimi
- 2-(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)-1-[2-[(1R)-5-(6-methylpyrimidin-4-yl)-2,3-dihydro-1H-inden-1-yl]-2,7-diaz...
- NBI 35965 hydrochloride◐ .Su ordinazione · 8–12 settimane Oggetto #: N288172Visualizza prodottoPrezzi e dimensioni del pacchetto
Identificatori tecnici
- Nome IUPAC
- (10S)-9-(cyclopropylmethyl)-3-(2,4-dichlorophenyl)-10-ethyl-6-methyl-1,2,5,9-tetrazatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraene;hydrochloride
- SMILES
- CCC1CN2C3=C(N1CC4CC4)C=C(N=C3C(=N2)C5=C(C=C(C=C5)Cl)Cl)C.Cl
- InChIKey
- LNYUWBPFYXPUIO-RSAXXLAASA-N
- InChI
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- Sinonimi
- 1782228-59-4 | DTXSID10849508 | (10S)-9-(cyclopropylmethyl)-3-(2,4-dichlorophenyl)-10-ethyl-6-methyl-1,2,5,9-tetrazat...
- GTS-21 dihydrochloride (DMBX-A)● In magazzino — Magazzino negli USA, spedizione nell'EU* Oggetto #: G275216Visualizza prodottoPrezzi e dimensioni del pacchetto
Identificatori tecnici
- Nome IUPAC
- 3-[(5E)-5-[(2,4-dimethoxyphenyl)methylidene]-3,4-dihydro-2H-pyridin-6-yl]pyridine;dihydrochloride
- SMILES
- COC1=CC(=C(C=C1)C=C2CCCN=C2C3=CN=CC=C3)OC.Cl.Cl
- InChIKey
- BXKYFUGAAFLYJL-BXGYHSFXSA-N
- InChI
- 1S/C19H20N2O2.2ClH/c1-22-17-8-7-14(18(12-17)23-2)11-15-5-4-10-21-19(15)16-6-3-9-20-13-16;;/h3,6-9,11-13H,4-5,10H2,1-2H3;2*1H/b15-11+;;
- Sinonimi
- AKOS037515500 | SCHEMBL8003 | DMXB | DANSYLAMIDE [FOR FLUOROMETRY] | Gts 21 | GTS-21 2HCl | GTS-21 (dihydrochloride) ...
- Luteinizing Hormone Releasing Hormone-III◐ .Su ordinazione · 8–12 settimane Oggetto #: L274664Visualizza prodottoPrezzi e dimensioni del pacchetto
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- Nome IUPAC
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- SMILES
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- InChIKey
- RTASYRSYWSLWJV-CSYZDTNESA-N
- InChI
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- Sinonimi
- LGnRH-III, lamprey | GnRH III | NCGC00167299-01 | GLYCINAMIDE, 5-OXO-L-PROLYL-L-HISTIDYL-L-TRYPTOPHYL-L-SERYL-L-HISTI...
- Luzindole, Antagonist of MT 1 receptor;Antagonist of MT 2 receptorCAS: 117946-91-5 Formula: C19H20N2O Peso molecolare: 292.37Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥96%● In magazzino — Magazzino negli USA, spedizione nell'EU* Oggetto #: L132758Visualizza prodottoPrezzi e dimensioni del pacchetto
Identificatori tecnici
- Nome IUPAC
- N-[2-(2-benzyl-1H-indol-3-yl)ethyl]acetamide
- SMILES
- CC(=O)NCCC1=C(NC2=CC=CC=C21)CC3=CC=CC=C3
- InChIKey
- WVVXBPKOIZGVNS-UHFFFAOYSA-N
- InChI
- 1S/C19H20N2O/c1-14(22)20-12-11-17-16-9-5-6-10-18(16)21-19(17)13-15-7-3-2-4-8-15/h2-10,21H,11-13H2,1H3,(H,20,22)
- Sinonimi
- 2-Benzyl-N-acetyltryptamine | HMS3411B10 | N-(2-(2-(PHENYLMETHYL)-1H-INDOL-3-YL)ETHYL)ETHANAMIDE | AM20020263 | Q6706...
- NF 157◐ .Su ordinazione · 8–12 settimane Oggetto #: N288559Visualizza prodottoPrezzi e dimensioni del pacchetto
Identificatori tecnici
- SMILES
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- InChIKey
- QJFCMJZVZFAWGF-UHFFFAOYSA-H
- Sinonimi
- NF 157 | AKOS024457107 | Hexasodium;8-[[4-fluoro-3-[[3-[[3-[[2-fluoro-5-[(8-oxidoperoxysulfanyl-4,6-disulfonatonaphth...
- PD 168077 maleateCAS: 630117-19-0 Formula: C20H22N4O.C4H4O4 Peso molecolare: 450.49● In magazzino — Magazzino negli USA, spedizione nell'EU* Oggetto #: P286721Visualizza prodottoPrezzi e dimensioni del pacchetto
Identificatori tecnici
- Nome IUPAC
- (Z)-but-2-enedioic acid;N-[[4-(2-cyanophenyl)piperazin-1-yl]methyl]-3-methylbenzamide
- SMILES
- CC1=CC(=CC=C1)C(=O)NCN2CCN(CC2)C3=CC=CC=C3C#N.C(=CC(=O)O)C(=O)O
- InChIKey
- NAEUGRPISCANHO-BTJKTKAUSA-N
- InChI
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- Sinonimi
- N-((4-(2-Cyanophenyl)-1-piperazinyl)methyl)-3-methylbenzamide (2Z)-2-butenedioate (1:1) | HY-21098A | N-(Methyl-4-(2-...
- GSK 789472 hydrochloride● In magazzino — Magazzino negli USA, spedizione nell'EU* Oggetto #: G344393Visualizza prodottoPrezzi e dimensioni del pacchetto
Identificatori tecnici
- Nome IUPAC
- 1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one;hydrochloride
- SMILES
- C1CCNC(C1)CN2CCN(C2=O)C3=CC=CC=C3.Cl
- InChIKey
- BYJUVPWUMBVSTK-UHFFFAOYSA-N
- InChI
- 1S/C15H21N3O.ClH/c19-15-17(12-13-6-4-5-9-16-13)10-11-18(15)14-7-2-1-3-8-14;/h1-3,7-8,13,16H,4-6,9-12H2;1H
- Sinonimi
- 1257326-24-1 | 1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one hydrochloride | GSK 789472 hydrochloride | MFCD180...
- NBI 27914 hydrochloride, Antagonist of CRF 1 receptorSolido Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥99%◐ .Su ordinazione · 8–12 settimane Oggetto #: N332118Visualizza prodottoPrezzi e dimensioni del pacchetto
Identificatori tecnici
- Nome IUPAC
- 5-chloro-4-N-(cyclopropylmethyl)-2-methyl-4-N-propyl-6-N-(2,4,6-trichlorophenyl)pyrimidine-4,6-diamine
- SMILES
- CCCN(CC1CC1)C2=NC(=NC(=C2Cl)NC3=C(C=C(C=C3Cl)Cl)Cl)C
- InChIKey
- KNADXBVKFAUMCR-UHFFFAOYSA-N
- InChI
- 1S/C18H20Cl4N4/c1-3-6-26(9-11-4-5-11)18-15(22)17(23-10(2)24-18)25-16-13(20)7-12(19)8-14(16)21/h7-8,11H,3-6,9H2,1-2H3,(H,23,24,25)
- Sinonimi
- CAS-29964-84-9 | NCGC00015737-04 | NCGC00015737-05 | NCGC00015737-08 | 4,6-Pyrimidinediamine, 5-chloro-N-(cyclopropyl...
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Domande frequenti
How do I choose the right GPCR/G Protein product for my experiment?
Match the GPCR/G Protein product to the application first — Western blot, ELISA, cell-based assay, and structural work make different demands. Then check species reactivity or source organism, format (lyophilised or solution), and whether you need an activity-verified lot.
What does the GPCR/G Protein category include?
GPCR/G Protein covers 5-HT Receptor, Adenosine Receptor, Adenylate Cyclase, Adrenergic Receptor and Amylin Receptor, and 76 further subcategories. Each product page lists format, purity, and storage so items from different subcategories can be compared on the same terms.
What specifications matter most for GPCR/G Protein?
For GPCR/G Protein, check purity by SDS-PAGE or HPLC, endotoxin level for cell-based work, specific activity, tag and expression system, and the reconstitution and storage conditions. Repeated freeze-thaw is the commonest cause of lost activity. All products are supplied for professional research and development use only, and are not for use in humans, animals, diagnostics, or therapy.
Can I search GPCR/G Protein by target, species, or application?
Yes — filter GPCR/G Protein by application, species reactivity or source, and format, and search by gene or protein name. For items not listed, contact [email protected]. We supply verified businesses, research institutions, universities, and government agencies.












