GRADE & PURITYMoligand™?Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools.10 mM in DMSO
Moligand™, 10 mM in DMSO Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
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Storage & shipping
Store at -80°C Ships Dry ice packs + Cold packs Check lot-specific COA for exact specifications.
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Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
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Literature proof
Cited in 1 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Overview
Amiloride (MK-870) is an inhibitor of both epithelial sodium channel ( ENaC) and urokinase-type plasminogen activator receptor ( uTPA). Amiloride is a blocker of polycystin-2 (PC2; TRPP2) channel.
Specifications
Specifications & Purity
Moligand™, 10 mM in DMSO
Storage
Store at -80°C
Shipped In
Dry ice packs + Cold packs
This product requires cold chain shipping. Ground and other economy services are not available.
Grade
Moligand™
Product Properties
pKa
pKa: 7.81 (Predicted), pKa: 3.78 (Predicted)
Ki Data
uPA: Ki= 2.51 μM (human); Adenosine A2A-R: Ki= 3.28 μM (human); Solute carrier family 22 member 2: Ki= 4.7 μM (rat); Solute carrier family 22 member 1: Ki= 6.9 μM (rat); Amine oxidase, copper containing: Ki= 10 μM (rat)
Names and Identifiers
Isomeric SMILES
C1(=C(N=C(C(=N1)Cl)N)N)C(=O)N=C(N)N
Alternate CAS
2016-88-8;17440-83-4
Molecular Weight
229.63
Beilstein
616612
Documentation
📋 Safety Data Sheet (SDS)
Comprehensive hazard, handling, storage, and regulatory compliance document.
1.Ruoning Wang, Qifan Liang, Xinru Zhang, Zhenning Di, Xiaohong Wang, Liuqing Di. (2022) Tumor-derived exosomes reversing TMZ resistance by synergistic drug delivery for glioma-targeting treatment. COLLOIDS AND SURFACES B-BIOINTERFACES, [PMID:35487070][10.1016/j.colsurfb.2022.112505]
Solution Calculators
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Reviews
Customer Reviews
Frequently Asked Questions
What is Moligand??
Moligand? is one of Aladdin Scientific's premium product lines, formulated for high-purity applications across multiple workflows. Compared to standard grades in the same workflow, Moligand? products typically offer tighter specifications, more rigorous QC, and stronger lot-to-lot consistency.
How should this product be stored?
Store at ?80 °C. Ultra-low temperature storage is required to maintain the specified shelf life.
How is this product shipped?
This product ships frozen with dry ice and cold packs. Unpack on arrival and transfer it to the storage condition stated above; handle dry ice with insulated gloves in a ventilated area.
What documentation is provided?
Available product documentation, including Certificates of Analysis (COA), Safety Data Sheets (SDS), and specification sheets, is shown in the product document area. Document availability and access follow the current site policy.
What are the CAS number, molecular formula and molecular weight?
The CAS Number is 2609-46-3, the molecular formula is C6H8ClN7O, and the molecular weight is 229.63 g/mol.
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