Azasetron HCl - ≥99% , CAS No.123040-16-4
In stock
SKU
A129701
Potent, selective, competitive 5-HT3 receptor antagonist with antiemetic effects
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Potent, selective, competitive 5-HT3 receptor antagonist with antiemetic effects
Azasetron HCl is a selective 5-HT3 receptor antagonist with IC50 of 0.33 nM used in the management of nausea and vomiting induced by cancer chemotherapy.
A potent and selective SR-3 antagonist
| CAS | 123040-16-4 |
|---|---|
| Synonyms | DTXSID00924358 | N-1-Azabicyclo[2.2.2]-oct-3-yl-6-chloro-3,4-dihydro-4-methyl-3-oxo-2H-1,4-benzoxazine-8-carboxamide Hydrochloride | (-)-6-Chloro-4-methyl-3-oxo-3,4-dihydro-2H-benzo[1,4]oxazine-8-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide hydroc |
| Specifications & Purity | ≥99% |
| Storage | Store at -20°C |
| Shipped In | Ice chest + Ice pads |
| Product Description | Azasetron HCl is a selective 5-HT3 receptor antagonist with IC50 of 0.33 nM used in the management of nausea and vomiting induced by cancer chemotherapy. |
| Pubchem Sid | 528776298 |
| Solubility | Soluble in water (25 mg/ml), and DMSO (10 mM). |
| Sensitivity | Hygroscopic |
| PubChem CID | 115000 |
| Molecular Formula | C17H21Cl2N3O3 |