GPCR/G Protein - GHSR Supplier | High Purity

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PF 05190457, Antagonist of ghrelin receptor
CAS: 1334782-79-4 PubChem CID: 58438464 Formula: C₂₉H₃₂N₆OS Molecular Weight: 512.67

Moligand™ ? ≥98%(HPLC)

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IUPAC Name

2-(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)-1-[2-[(1R)-5-(6-methylpyrimidin-4-yl)-2,3-dihydro-1H-inden-1-yl]-2,7-diazaspiro[3.5]nonan-7-yl]ethanone

SMILES

CC1=CC(=NC=N1)C2=CC3=C(C=C2)C(CC3)N4CC5(C4)CCN(CC5)C(=O)CC6=CN7C=C(SC7=N6)C

InChIKey
ZIUDADZJCKGWKR-AREMUKBSSA-N

InChI

1S/C29H32N6OS/c1-19-11-25(31-18-30-19)22-3-5-24-21(12-22)4-6-26(24)35-16-29(17-35)7-9-33(10-8-29)27(36)13-23-15-34-14-20(2)37-28(34)32-23/h3,5,11-12,1show more

Synonyms
2-(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)-1-[2-[(1R)-5-(6-methylpyrimidin-4-yl)-2,3-dihydro-1H-inden-1-yl]-2,7-diaz...
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PF 04628935
CAS: 1383719-97-8 PubChem CID: 70682037 Formula: C₂₄H₂₆ClN₇OS Molecular Weight: 496.03

≥98%(HPLC)

◐ .Made to order · 8–12 wks Item #: P288177
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IUPAC Name

1-[2-[[2-chloro-4-(triazol-2-yl)phenyl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)ethanone

SMILES

CC1=CN2C=C(N=C2S1)CC(=O)N3CCC4(CC3)CN(C4)CC5=C(C=C(C=C5)N6N=CC=N6)Cl

InChIKey
MTDYDDJVCIHZKH-UHFFFAOYSA-N

InChI

1S/C24H26ClN7OS/c1-17-12-31-14-19(28-23(31)34-17)10-22(33)30-8-4-24(5-9-30)15-29(16-24)13-18-2-3-20(11-21(18)25)32-26-6-7-27-32/h2-3,6-7,11-12,14H,4-5show more

Synonyms
1-[2-[[2-Chloro-4-(2H-1,2,3-triazol-2-yl)phenyl]methyl]-2,7-diazaspiro[3.5]non-7-yl]-2-(2-methylimidazo[2,1-b]thiazol...
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YIL 781 hydrochloride
CAS: 1640226-17-0 PubChem CID: 74889155 Formula: C₂₄H₂₉ClFN₃O₂ Molecular Weight: 445.96

≥98%(HPLC)

◐ .Made to order · 8–12 wks Item #: Y287105
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IUPAC Name

6-(4-fluorophenoxy)-2-methyl-3-[[(3S)-1-propan-2-ylpiperidin-3-yl]methyl]quinazolin-4-one;hydrochloride

SMILES

CC1=NC2=C(C=C(C=C2)OC3=CC=C(C=C3)F)C(=O)N1CC4CCCN(C4)C(C)C.Cl

InChIKey
QQGRMONBDBMLSP-FERBBOLQSA-N

InChI

1S/C24H28FN3O2.ClH/c1-16(2)27-12-4-5-18(14-27)15-28-17(3)26-23-11-10-21(13-22(23)24(28)29)30-20-8-6-19(25)7-9-20;/h6-11,13,16,18H,4-5,12,14-15H2,1-3H3show more

Synonyms
YIL781 HCl | YIL 781 HCl | 6-(4-Fluorophenoxy)-2-methyl-3-[[(3S)-1-(1-methylethyl)-3-piperidinyl]methyl]-4(3H)-quinaz...
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MK 0677
CAS: 159752-10-0 PubChem CID: 6450830 Formula: C₂₈H₄₀N₄O₈S₂ Molecular Weight: 624.77

Solid Moligand™ ? ≥98%(HPLC)

● In Stock — US warehouse, ships to EU* Item #: M288146
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IUPAC Name

2-amino-2-methyl-N-[(2R)-1-(1-methylsulfonylspiro[2H-indole-3,4'-piperidine]-1'-yl)-1-oxo-3-phenylmethoxypropan-2-yl]propanamide;methanesulfonic acid

SMILES

CC(C)(C(=O)NC(COCC1=CC=CC=C1)C(=O)N2CCC3(CC2)CN(C4=CC=CC=C34)S(=O)(=O)C)N.CS(=O)(=O)O

InChIKey
DUGMCDWNXXFHDE-VZYDHVRKSA-N

InChI

1S/C27H36N4O5S.CH4O3S/c1-26(2,28)25(33)29-22(18-36-17-20-9-5-4-6-10-20)24(32)30-15-13-27(14-16-30)19-31(37(3,34)35)23-12-8-7-11-21(23)27;1-5(2,3)4/h4-show more

Synonyms
2-amino-2-methyl-N-[(2R)-1-(1-methylsulfonylspiro[2H-indole-3,4'-piperidine]-1'-yl)-1-oxo-3-phenylmethoxypropan-2-yl]...
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Anamorelin
CAS: 249921-19-5 Formula: C₃₁H₄₂N₆O₃ Molecular Weight: 546.7

≥98%

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IUPAC Name

2-amino-N-[(2R)-1-[(3R)-3-benzyl-3-[dimethylamino(methyl)carbamoyl]piperidin-1-yl]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-methylpropanamide

SMILES

CC(C)(C(=O)NC(CC1=CNC2=CC=CC=C21)C(=O)N3CCCC(C3)(CC4=CC=CC=C4)C(=O)N(C)N(C)C)N

InChIKey
VQPFSIRUEPQQPP-MXBOTTGLSA-N

InChI

1S/C31H42N6O3/c1-30(2,32)28(39)34-26(18-23-20-33-25-15-10-9-14-24(23)25)27(38)37-17-11-16-31(21-37,29(40)36(5)35(3)4)19-22-12-7-6-8-13-22/h6-10,12-15,show more

Synonyms
RC-1291 | CCG-269985 | UNII-6MUC9717YK | HY-14734 | RC-1291;ONO-7643 | ST-1291 | UNII-DD5RBA1NKF | Q20707542 | RC-129...
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TC-G 1008
CAS: 1621175-65-2 PubChem CID: 91826086 Formula: C₁₈H₁₉ClN₆O₂S Molecular Weight: 418.9

≥98%(HPLC)

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IUPAC Name

N-[3-chloro-4-[[[2-(methylamino)-6-pyridin-2-ylpyrimidin-4-yl]amino]methyl]phenyl]methanesulfonamide

SMILES

CNC1=NC(=CC(=N1)NCC2=C(C=C(C=C2)NS(=O)(=O)C)Cl)C3=CC=CC=N3

InChIKey
DRSZMILOMUPIBJ-UHFFFAOYSA-N

InChI

1S/C18H19ClN6O2S/c1-20-18-23-16(15-5-3-4-8-21-15)10-17(24-18)22-11-12-6-7-13(9-14(12)19)25-28(2,26)27/h3-10,25H,11H2,1-2H3,(H2,20,22,23,24)

Synonyms
GPR39-C3 | N-[3-Chloro-4-[[[2-(methylamino)-6-(2-pyridinyl)-4-pyrimidinyl]amino]methyl]phenyl]methanesulfonamide | TC...
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GHRF (1-44), human GRF, Agonist of GHRH receptor;Agonist of VPAC 1 receptor
CAS: 83930-13-6 PubChem CID: 16132353 Formula: C₂₁₅H₃₅₈N₇₂O₆₆S Molecular Weight: 5039.65

Moligand™ ? ≥95%(HPLC)

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IUPAC Name

(4S)-4-[[2-[[(2S)-5-amino-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2Sshow more

SMILES

CCC(C)C(C(=O)NC(CC1=CC=CC=C1)C(=O)NC(C(C)O)C(=O)NC(CC(=O)N)C(=O)NC(CO)C(=O)NC(CC2=CC=C(C=C2)O)C(=O)NC(CCCNC(=N)N)C(=O)NC(CCCCN)C(=O)NC(C(C)C)C(=O)NC(Cshow more

InChIKey
JAHCMOSSKRAPEL-IBFVROBCSA-N

InChI

1S/C215H358N72O66S/c1-24-106(15)166(285-174(318)112(21)251-193(337)145(91-163(309)310)270-173(317)109(18)249-175(319)119(218)86-115-49-53-117(293)54-5show more

Synonyms
UNII-4UR7N9Z9MM | Somatorelin | DTXSID40232828 | PD151144 | 4UR7N9Z9MM | GRF (1-44), human | Somatorelin [INN]
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TM N1324
CAS: 1144477-35-9 PubChem CID: 135634901 Formula: C₁₈H₁₃ClFN₇O Molecular Weight: 397.79

≥98%(HPLC)

◐ .Made to order · 8–12 wks Item #: T287495
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IUPAC Name

4-(2-chloro-4-fluorophenyl)-3-methyl-1-(7H-purin-6-yl)-5,7-dihydro-4H-pyrazolo[3,4-b]pyridin-6-one

SMILES

CC1=NN(C2=C1C(CC(=O)N2)C3=C(C=C(C=C3)F)Cl)C4=NC=NC5=C4NC=N5

InChIKey
CYQNVXRIWKKWQG-UHFFFAOYSA-N

InChI

1S/C18H13ClFN7O/c1-8-14-11(10-3-2-9(20)4-12(10)19)5-13(28)25-17(14)27(26-8)18-15-16(22-6-21-15)23-7-24-18/h2-4,6-7,11H,5H2,1H3,(H,25,28)(H,21,22,23,24show more

Synonyms
4-(2-Chloro-4-fluorophenyl)-1,4,5,7-tetrahydro-3-methyl-1-(9H-purin-6-yl)-6H-pyrazolo[3,4-b]pyridin-6-one
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Obestatin human(trifluoroacetate salt)
CAS: 1081110-72-6 PubChem CID: 146156385 Formula: C₁₁₆H₁₇₆N₃₂O₃₃（free basis） Molecular Weight: 2546.86（free basis）

≥95%

● In Stock — US warehouse, ships to EU* Item #: O287703
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IUPAC Name

4-[[1-[[2-[[1-[[6-amino-1-[[1-[[1-[[2-[[1-[[5-amino-1-[[1-[[5-amino-1-[[5-amino-1-[[1-[[1-[[5-amino-1-[[1-[(1-amino-4-methyl-1-oxopentan-2-yl)amino]-1show more

SMILES

CCC(C)C(C(=O)NC(CCCCN)C(=O)NC(CC(C)C)C(=O)NC(CO)C(=O)NCC(=O)NC(C(C)C)C(=O)NC(CCC(=O)N)C(=O)NC(CC1=CC=C(C=C1)O)C(=O)NC(CCC(=O)N)C(=O)NC(CCC(=O)N)C(=O)Nshow more

InChIKey
IXQOGPZNKNSCJR-UHFFFAOYSA-N

InChI

1S/C116H176N32O33/c1-13-61(10)95(146-91(158)53-127-113(178)93(59(6)7)147-110(175)81(50-92(159)160)141-108(173)78(46-65-25-18-15-19-26-65)142-112(177)8show more
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Anamorelin
CAS: 249921-19-5 EC Number: 111-195-8 Formula: C₃₁H₄₂N₆O₃ Molecular Weight: 546.7

10mM in DMSO

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IUPAC Name

2-amino-N-[(2R)-1-[(3R)-3-benzyl-3-[dimethylamino(methyl)carbamoyl]piperidin-1-yl]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-2-methylpropanamide

SMILES

CC(C)(C(=O)NC(CC1=CNC2=CC=CC=C21)C(=O)N3CCCC(C3)(CC4=CC=CC=C4)C(=O)N(C)N(C)C)N

InChIKey
VQPFSIRUEPQQPP-MXBOTTGLSA-N

InChI

1S/C31H42N6O3/c1-30(2,32)28(39)34-26(18-23-20-33-25-15-10-9-14-24(23)25)27(38)37-17-11-16-31(21-37,29(40)36(5)35(3)4)19-22-12-7-6-8-13-22/h6-10,12-15,show more

Synonyms
RC-1291 | CCG-269985 | UNII-6MUC9717YK | HY-14734 | RC-1291;ONO-7643 | ST-1291 | UNII-DD5RBA1NKF | Q20707542 | RC-129...
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Capromorelin tartrate
CAS: 193273-69-7 EC Number: 110-650-8 PubChem CID: 9852610 Formula: C₃₂H₄₁N₅O₁₀ Molecular Weight: 655.7

10mM in DMSO

● In Stock — US warehouse, ships to EU* Item #: C422360
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IUPAC Name

N-[(2R)-1-[(3aR)-3a-benzyl-2-methyl-3-oxo-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]-1-oxo-3-phenylmethoxypropan-2-yl]-2-amino-2-methylpropanamide;(2show more

SMILES

CC(C)(C(=O)NC(COCC1=CC=CC=C1)C(=O)N2CCC3=NN(C(=O)C3(C2)CC4=CC=CC=C4)C)N.C(C(C(=O)O)O)(C(=O)O)O

InChIKey
MJGRJCMGMFLOET-MYPSAZMDSA-N

InChI

1S/C28H35N5O4.C4H6O6/c1-27(2,29)25(35)30-22(18-37-17-21-12-8-5-9-13-21)24(34)33-15-14-23-28(19-33,26(36)32(3)31-23)16-20-10-6-4-7-11-20;5-1(3(7)8)2(6)show more

Synonyms
193273-69-7 (tartrate) | Capromorelin tartrate [USAN] | D03373 | PROPANAMIDE, 2-AMINO-N-(2-(2,3,3A,4,6,7-HEXAHYDRO-2-...
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Capromorelin tartrate
CAS: 193273-69-7 PubChem CID: 9852610 Formula: C₃₂H₄₁N₅O₁₀ Molecular Weight: 655.7

≥95%

● In Stock — US warehouse, ships to EU* Item #: C412217
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IUPAC Name

N-[(2R)-1-[(3aR)-3a-benzyl-2-methyl-3-oxo-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]-1-oxo-3-phenylmethoxypropan-2-yl]-2-amino-2-methylpropanamide;(2show more

SMILES

CC(C)(C(=O)NC(COCC1=CC=CC=C1)C(=O)N2CCC3=NN(C(=O)C3(C2)CC4=CC=CC=C4)C)N.C(C(C(=O)O)O)(C(=O)O)O

InChIKey
MJGRJCMGMFLOET-MYPSAZMDSA-N

InChI

1S/C28H35N5O4.C4H6O6/c1-27(2,29)25(35)30-22(18-37-17-21-12-8-5-9-13-21)24(34)33-15-14-23-28(19-33,26(36)32(3)31-23)16-20-10-6-4-7-11-20;5-1(3(7)8)2(6)show more

Synonyms
193273-69-7 (tartrate) | Capromorelin tartrate [USAN] | D03373 | PROPANAMIDE, 2-AMINO-N-(2-(2,3,3A,4,6,7-HEXAHYDRO-2-...

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Frequently Asked Questions

How is the GHSR listing put together?

It draws on reported GHSR annotations within GPCR/G Protein and lists each compound with its structure, identifiers, and the activity published for it. Always check the underlying assay before comparing potency values across entries.

How do I choose a GHSR modulator for my assay?

Start from the assay format and readout — biochemical, cell-based, or in vivo — then compare the GHSR entries on potency, selectivity over related family members, and solubility in your vehicle. Where several chemotypes are available, a reference compound plus a structurally unrelated backup is the usual way to control for off-target effects.

Which specifications matter most for GHSR compounds?

Purity and identity confirmation come first, then solubility in DMSO or your chosen vehicle, recommended storage temperature, and stability in solution. For GHSR work in particular, freshly prepared stocks avoid most of the reproducibility problems seen with stored plates. All products are supplied for professional research and development use only, and are not for use in humans, animals, diagnostics, or therapy.

What if the GHSR compound I need is not listed?

Search by CAS number or SMILES first, since analogs of GHSR compounds are often catalogued under a related target. Custom synthesis and bulk enquiries go to [email protected]. We supply verified businesses, research institutions, universities, and government agencies.