DCLX069 - ≥98% , CAS No.792946-69-1

CAS: 792946-69-1 Cat. No.: D650930 Formula: C₂₀H₂₅N₃O₂ Molecular Weight: 339.43

GRADE & PURITY ≥98%

Storage

Protected from light,Store at -80°C

Shipped In

Dry ice packs + Cold packs

Overview

DCLX069 is a selective protein arginine methyltransferase 1 (PRMT1) inhibitor with an IC 50 value of 17.9 µM. DCLX069 shows less active against PRMT4 and PRMT6 . DCLX069 has anticancer effects

In Vitro

DCLX069 (12.5-100 µM) effectively blocks cell proliferation in breast cancer, liver cancer and acute myeloid leukemia cell lines (MCF7, HepG2, and THP1 cells) in a concentration-dependent manner. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Form:Solid

IC50& Target:PRMT1 17.9 μM (IC 50 )

Specifications

Specifications & Purity

≥98%

Biochemical and Physiological Mechanisms

DCLX069 is a selective protein arginine methyltransferase 1 (PRMT1) inhibitor with an IC 50 value of 17.9 µM. DCLX069 shows less active against PRMT4 and PRMT6 . DCLX069 has anticancer effects.

Storage

Protected from light,Store at -80°C

Shipped In

Dry ice packs + Cold packs

This product requires cold chain shipping. Ground and other economy services are not available.

Action Type

INHIBITOR

Purity

≥98%

Names and Identifiers

• Molecular Weight: 339.43

Chemical and Physical Properties

• Solubility: DMSO : 100 mg/mL (294.61 mM; Need ultrasonic)