Enpp-1-IN-2 - ≥99% , CAS No.2378640-92-5

CAS: 2378640-92-5 Cat. No.: E650422 Molecular Weight: 282.34 PubChem CID: 156589002

GRADE & PURITY ≥99%

Synonyms

Enpp-1-IN-2 | 6-[(3-aminophenyl)methyl]-N,N,5-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine | ENPP1 Inhibitor C | SCHEMBL24129143 | AKOS040755821 | MS-24013 | HY-139362 | Z4180066045

Storage

Store at -20°C

Shipped In

Ice chest + Ice pads

Overview

Enpp-1-IN-2 (Compound C) is a potent ENPP1 (ectonucleotide pyrophosphatase/phosphodiesterase 1) inhibitor with IC 50 values of 0.26, 0.48 and 2.0 μM evaluated by means of TG-mAMP, pNP-TMP, and ATP assays, respectively. TG (Tokyo Green)-mAMP: a newly synthesized sensitive ENPP1 fluorescence probe

Form:Solid

IC50& Target:IC 50 : 0.26 μM (TG-mAMP assay), 0.48 μM (pNP-TMP assay), 2.0 μM (ATP assay)

Specifications

Synonyms

Enpp-1-IN-2 | 6-[(3-aminophenyl)methyl]-N, N, 5-trimethyl-[1, 2, 4]triazolo[1, 5-a]pyrimidin-7-amine | ENPP1 Inhibitor C | SCHEMBL24129143 | AKOS040755821 | MS-24013 | HY-139362 | Z4180066045

Specifications & Purity

≥99%

Biochemical and Physiological Mechanisms

Enpp-1-IN-2 (Compound C) is a potent ENPP1 (ectonucleotide pyrophosphatase/phosphodiesterase 1) inhibitor with IC 50 values of 0.26, 0.48 and 2.0 μM evaluated by means of TG-mAMP, pNP-TMP, and ATP assays, respectively. TG (Tokyo Green)-mAMP: a newly synth

Storage

Store at -20°C

Shipped In

Ice chest + Ice pads

This product requires cold chain shipping. Ground and other economy services are not available.

Action Type

INHIBITOR

Purity

≥99%

Names and Identifiers

• Canonical Smiles: CC1=NC2=NC=NN2C(=C1CC3=CC(=CC=C3)N)N(C)C
• IUPAC Name: 6-[(3-aminophenyl)methyl]-N,N,5-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
• InChIKey: VUDSCOCEYOZLJD-UHFFFAOYSA-N
• INCHI: 1S/C15H18N6/c1-10-13(8-11-5-4-6-12(16)7-11)14(20(2)3)21-15(19-10)17-9-18-21/h4-7,9H,8,16H2,1-3H3
• PubChem CID: 156589002
• Molecular Weight: 282.34