LDN-57444 - ≥98%(HPLC) , CAS No.668467-91-2
In stock
SKU
L137664
Reversible, competitive UCH-L1 inhibitor
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Reversible, competitive UCH-L1 inhibitor
LDN-57444 is a reversible, competitive proteasome inhibitor for Uch-L1 with IC50 of 0.88 μM, 28-fold selectivity over isoform Uch-L3.
A potent, reversible, active site-directed UCH-L1 inhibitor
| CAS | 668467-91-2 |
|---|---|
| Synonyms | HY-18637 | SW219408-1 | UCH-L1 | [(Z)-[5-chloro-1-[(2,5-dichlorophenyl)methyl]-2-oxoindol-3-ylidene]amino] acetate | LDN 57444 | SCHEMBL16249746 | 5-Chloro-1-[(2,5-dichlorophenyl)methyl]-1H-indole-2,3-dione 3-(O-acetyloxime) | LDN-57444, >=98% (HPLC) | BD |
| Specifications & Purity | ≥98%(HPLC) |
| Storage | Store at 2-8°C |
| Shipped In | Wet ice |
| Product Description | LDN-57444 is a reversible, competitive proteasome inhibitor for Uch-L1 with IC50 of 0.88 μM, 28-fold selectivity over isoform Uch-L3. |
| Pubchem Sid | 508810698 |
| Solubility | Soluble in DMSO (20 mg/ml). |
| Target | UCHL1 |
| Mdl Number | MFCD09037562 |
| PubChem CID | 16760696 |
| Molecular Formula | C17H11Cl3N2O3 |