LP-922761 - Moligand™, 10 mM in DMSO , CAS No.1454808-95-7
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SKU
L1495260
LP-922761 is a potent, selective and orally active adapter protein-2 associated kinase 1 ( AAK1 ) inhibitor with IC 50 s of 4.8 nM and 7.6 nM in enzyme and cell assays, respectively.LP-922761 also inhibits BMP-2-inducible protein kinase (BIKE) with an IC 50 of 24 nM. LP-922761 exhibits no significant activity at cyclin G-associated kinase (GAK) , opioid, adrenergic α2 or GABAa receptors.
More Information
| CAS | 1454808-95-7 |
|---|---|
| Concentration | 10 mM in DMSO |
| Specifications & Purity | Moligand™, 10 mM in DMSO |
| Storage | Store at -80°C |
| Shipped In | Dry ice packs + Cold packs |
| Product Description | LP-922761 is a potent, selective and orally active adapter protein-2 associated kinase 1 ( AAK1 ) inhibitor with IC 50 s of 4.8 nM and 7.6 nM in enzyme and cell assays, respectively.LP-922761 also inhibits BMP-2-inducible protein kinase (BIKE) with an IC 50 of 24 nM. LP-922761 exhibits no significant activity at cyclin G-associated kinase (GAK) , opioid, adrenergic α2 or GABAa receptors. |
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