Rebamipide - Moligand™, 10mM in DMSO , Agonist of CCK 1 receptor, CAS No.90098-04-7, Agonist of CCK 1 receptor

CAS: 90098-04-7 Cat. No.: R408057 Formula: C₁₉H₁₅ClN₂O₄.xH₂O Molecular Weight: 370.79 EC Number: 815-380-0 PubChem CID: 5042

GRADE & PURITY Moligand™, 10mM in DMSO

Synonyms

OPC-12759 | α-​[(4-​chlorobenzoyl)​amino]​-​1,​2-​dihydro-​2-​oxo-4-​quinolinepropanoic acid

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

Overview

Information

Rebamipide Rebamipide (OPC-12759) is a cholecystokinin type 1 (CCK1) receptor inhibitor for inhibiting [ 125 I]BH-CCK-8S with IC50 of 37.7 μM.
In vitro

In vivo

Cell Data

cell lines：

Concentrations：

Incubation Time：

Powder Purity:≥99%

Specifications

Synonyms

OPC-12759 | α-​[(4-​chlorobenzoyl)​amino]​-​1,​2-​dihydro-​2-​oxo-4-​quinolinepropanoic acid

Specifications & Purity

Moligand™, 10mM in DMSO

Biochemical and Physiological Mechanisms

Rebamipide (OPC-12759) is a cholecystokinin type 1 (CCK1) receptor inhibitor for inhibiting [¹²⁵I]BH-CCK-8S with IC50 of 37.7 μM.

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

This product requires cold chain shipping. Ground and other economy services are not available.

Grade

Moligand™

Action Type

AGONIST

Mechanism of action

Agonist of CCK 1 receptor

Names and Identifiers

• Isomeric SMILES: C1=CC=C2C(=C1)C(=CC(=O)N2)CC(C(=O)O)NC(=O)C3=CC=C(C=C3)Cl
• RTECS: VC2518500
• PubChem CID: 5042
• Molecular Weight: 370.79
• Reaxy-Rn: 5384689

Associated Targets(Human)

CCKAR Tclin Cholecystokinin receptor type A (1 Activities)

Discover Target: CCKAR

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Chemical and Physical Properties

• Melt Point(°C): 290°C(dec.)(lit.)

References

1. Han Qiao, Zhuo Xu, Mengchi Sun, Shuwen Fu, Fangxue Zhao, Danping Wang, Zhonggui He, Yinglei Zhai, Jin Sun.  (2022)  Rebamipide liposome as an effective ocular delivery system for the management of dry eye disease.  JOURNAL OF DRUG DELIVERY SCIENCE AND TECHNOLOGY,      [PMID:] [10.1016/j.jddst.2022.103654]