S961 TFA , CAS No.S659083

CAS: S659083 Cat. No.: S659083 Formula: C₂₁₁H₂₉₇N₅₅O₇₁S₂.C₂HF₃O₂ Molecular Weight: 4918.15

Storage

Protected from light,Desiccated,Store at -80°C

Shipped In

Dry ice packs + Cold packs

Overview

S961 TFA is an high-affinity and selective insulin receptor ( IR ) antagonist with IC 50 s of 0.048, 0.027, and 630 nM for HIR-A, HIR-B, and human insulin-like growth factor I receptor (HIGF-IR) in SPA-assay, respectively.

Appearance:Solid

In Vitro:S961 also shows high-affinity to Rat IR and Pig IR with IC 50 s of 0.056 nM and 0.084 nM in PEG-assay, respectively. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Biological Activity:S961 TFA is an high-affinity and selective insulin receptor ( IR ) antagonist with IC 50 s of 0.048, 0.027, and 630 nM for HIR-A, HIR-B, and human insulin-like growth factor I receptor (HIGF-IR) in SPA-assay, respectively.

Specifications

Storage

Protected from light,Desiccated,Store at -80°C

Shipped In

Dry ice packs + Cold packs

This product requires cold chain shipping. Ground and other economy services are not available.

Names and Identifiers

Molecular Weight

4918.15

Chemical and Physical Properties

• Solubility: H2O : 6.5 mg/mL (1.32 mM; ultrasonic and adjust pH to 12 with NaOH)