SKLB-03220 - Moligand™, ≥98% , Inhibitor of enhancer of zeste 2 polycomb repressive complex 2 subunit, CAS No.S613615, Inhibitor of enhancer of zeste 2 polycomb repressive complex 2 subunit

CAS: S613615 Cat. No.: S613615 Formula: C₃₃H₄₀N₄O₄ Molecular Weight: 556.7

GRADE & PURITY Moligand™, ≥98%

Synonyms

5'-Acrylamido-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-2',4-dimethyl-[1,1'-biphenyl]-3-carboxamide | GTPL12353 | GLXC-26853 | BDBM50616852

Storage

Store at -20°C

Shipped In

Ice chest + Ice pads

Specifications

Synonyms

5'-Acrylamido-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-2',4-dimethyl-[1,1'-biphenyl]-3-carboxamide | GTPL12353 | GLXC-26853 | BDBM50616852

Specifications & Purity

Moligand™, ≥98%

Storage

Store at -20°C

Shipped In

Ice chest + Ice pads

This product requires cold chain shipping. Ground and other economy services are not available.

Grade

Moligand™

Action Type

INHIBITOR

Mechanism of action

Inhibitor of enhancer of zeste 2 polycomb repressive complex 2 subunit

Purity

≥98%

Names and Identifiers

• Canonical Smiles: O=C(NCc1c(C)cc(C)[nH]c1=O)c1c(C)c(N(CC)C2CCOCC2)cc(c2cc(NC(=O)C=C)ccc2C)c1
• IUPAC Name: 5′-Acrylamido-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-2′,4-dimethyl-[1,1′-biphenyl]-3-carboxamide
• InChIKey: QKOGMESAENVJHH-UHFFFAOYSA-N
• INCHI: 1S/C33H40N4O4/c1-7-31(38)36-25-10-9-20(3)27(18-25)24-16-28(32(39)34-19-29-21(4)15-22(5)35-33(29)40)23(6)30(17-24)37(8-2)26-11-13-41-14-12-26/h7,9-10,15-18,26H,1,8,11-14,19H2,2-6H3,(H,34,39)(H,35,40)(H,36,38)
• Molecular Weight: 556.7

Associated Targets(Human)

EZH2 Tclin Histone-lysine N-methyltransferase EZH2 (0 Activities)

Discover Target: EZH2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)