Phenylbutazone - Moligand™, 10mM in DMSO , Inhibitor of COX-1;Inhibitor of COX-2, CAS No.50-33-9, Inhibitor of COX-1;Inhibitor of COX-2

CAS: 50-33-9 Cat. No.: P408411 Fórmula: C₁₉H₂₀N₂O₂ Peso molecular: 308.37 Beilstein Registry Number: 24(5)5,400 Número CE: 200-029-0

GRADE & PURITY Moligand™, 10mM in DMSO

Synonyms

Butazolidine | 4-​butyl-​1,​2-​diphenyl-3,​5-​pyrazolidinedione

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

Visão geral

Information

Phenylbutazone Phenylbutazone (Butazolidine) is used as a non-steroidal anti-inflammatory agent for the treatment of chronic pain, including the symptoms of arthritis.
In vitro

In vivo

Cell Data

cell lines：

Concentrations：

Incubation Time：

Powder Purity:≥100%

Specifications

Sinónimos

Butazolidine | 4-​butyl-​1,​2-​diphenyl-3,​5-​pyrazolidinedione

Especificações e pureza

Moligand™, 10mM in DMSO

Mecanismos bioquímicos e fisiológicos

Phenylbutazone (Butazolidine) is used as a non-steroidal anti-inflammatory agent for the treatment of chronic pain, including the symptoms of arthritis.

Condições de armazenamento de armazenamento

Store at -80°C

Enviado em

Dry ice packs + Cold packs

Este produto requer transporte de cadeia fria. Serviços terrestres e outros serviços econômicos não estão disponíveis.

Grau

Moligand™

Tipo de ação

INHIBITOR

Mecanismo de ação

Inhibitor of COX-1;Inhibitor of COX-2

Nomes e identificadores

• SMILES isoméricas: CCCCC1C(=O)N(N(C1=O)C2=CC=CC=C2)C3=CC=CC=C3
• WGK Alemanha: 3
• RTECS: UQ8225000
• Número UN: 2811
• Grupo de embalagem: I
• Peso molecular: 308.37
• Beilstein: 24(5)5,400
• Reaxy-Rn: 290080
• Reaxys-RN_link_address: https://www.reaxys.com/reaxys/secured/hopinto.do?context=S&query=IDE.XRN=290080&ln=

Alvos associados (humanos)

NAPRT Tchem Nicotinate phosphoribosyltransferase (2 Activities)

Discover Target: NAPRT

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

PTGS1 Tclin Prostaglandin G/H synthase 1 (1 Activities)

Discover Target: PTGS1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

PTGS2 Tclin Prostaglandin G/H synthase 2 (1 Activities)

Discover Target: PTGS2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Propriedades químicas e físicas

• Ponto de fusão (°C): 106 °C

Referências

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