TPMPA - Moligand™, ≥98%(HPLC) , Antagonist of GABA A receptor ρ1 subunit;Antagonist of GABA A receptor ρ2 subunit;Antagonist of GABA A receptor ρ3 subunit, CAS No.182485-36-5, Antagonist of GABA A receptor ρ1 subunit;Antagonist of GABA A receptor ρ2 subunit;Antagonist of GABA A receptor ρ3 subunit
TPMPA - Moligand™, ≥98%(HPLC) , Antagonist of GABA A receptor ρ1 subunit;Antagonist of GABA A receptor ρ2 subunit;Antagonist of GABA A receptor ρ3 subunit, CAS No.182485-36-5, Antagonist of GABA A receptor ρ1 subunit;Antagonist of GABA A receptor ρ2 subunit;Antagonist of GABA A receptor ρ3 subunit
GRAU & PUREZAMoligand™?Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools.≥98%(HPLC)
A selective, competitive GABAA-ρantagonist with only minimal effects on GABAAand GABABreceptors (Kbvalues are 2.1μM (antagonist), 320μM (antagonist) and EC50~ 500μM (weak agonist) respectively). Displays 8-fold selectivity for human recombinantρ1 receptor
Condições de armazenamento de armazenamento
Room temperature
Enviado em
Normal
Grau
Moligand™
Tipo de ação
ANTAGONIST
Mecanismo de ação
Antagonist of GABA A receptor ρ1 subunit;Antagonist of GABA A receptor ρ2 subunit;Antagonist of GABA A receptor ρ3 subunit
This compound belongs to the class of organic compounds known as hydropyridines. These are compounds containing a hydrogenated pyridine ring (i.e. containing less than the maximum number of double bonds.).
External Descriptors
Not available
1. Djoumbou Feunang Y, Eisner R, Knox C, Chepelev L, Hastings J, Owen G, Fahy E, Steinbeck C, Subramanian S, Bolton E, Greiner R, and Wishart DS. ClassyFire: Automated Chemical Classification With A Comprehensive, Computable Taxonomy. Journal of Cheminformatics, 2016, 8:61.
Solvent:water, Max Conc. mg/mL: None, Max Conc. mM: 100
Peso molecular
161.140 g/mol
XLogP3
-3.500
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
3
Rotatable Bond Count
1
Exact Mass
161.061 Da
Monoisotopic Mass
161.061 Da
Topological Polar Surface Area
49.300 Ų
Heavy Atom Count
10
Formal Charge
0
Complexity
200.000
Isotope Atom Count
0
Defined Atom Stereocenter Count
0
Undefined Atom Stereocenter Count
0
Defined Bond Stereocenter Count
0
Undefined Bond Stereocenter Count
0
The total count of all stereochemical bonds
0
Covalently-Bonded Unit Count
1
Calculadoras de soluções
Molarity Calculator
Determine the necessary mass, volume, or concentration for preparing a solution.
Dilution Calculator
Determine the dilution needed to prepare a stock solution.
Reconstitution Calculator
Revisões
Avaliações dos Clientes
Perguntas frequentes
What is the purity of this product, and how is it determined?
This product is supplied at ≥98% purity, determined by HPLC. Lot-specific values are stated on the Certificate of Analysis.
How should this product be stored?
Store at room temperature.
What is Moligand??
Moligand? is one of Aladdin Scientific's premium product lines, formulated for high-purity applications across multiple workflows. Compared to standard grades in the same workflow, Moligand? products typically offer tighter specifications, more rigorous QC, and stronger lot-to-lot consistency.
How is this product shipped?
This product ships under standard ambient conditions. No temperature-controlled packaging is required.
What are the CAS number, molecular formula and molecular weight?
The CAS Number is 182485-36-5, the molecular formula is C?H??NO?P, and the molecular weight is 161.14 g/mol. InChIKey MFUKVPOVVKKLRQ-UHFFFAOYSA-N.
What documentation is provided?
Available product documentation, including Certificates of Analysis (COA), Safety Data Sheets (SDS), and specification sheets, is shown in the product document area. Document availability and access follow the current site policy.
Precisa de ajuda para escolher o grau?
O nosso guia de seleção de graus abrange pureza, estado do estabilizador e adequação à aplicação para todas as variantes do nosso catálogo.
Usamos cookies para garantir o funcionamento adequado do site e, quando permitido, para melhorar a sua experiência. Você pode gerenciar suas preferências a qualquer momento nas Configurações. Saiba mais em nossa Política de Cookies.
Deseja que lhe enviemos uma mensagem quando tivermos descontos disponíveis?
Lembrar-me mais tarde
Obrigado! Por favor, verifique a sua caixa de entrada de e-mail para confirmar.
Products are supplied to verified businesses, institutions, and qualified professionals for research and development use only. Not for use in humans, animals, diagnosis, or therapy.
