γ1-MSH TFA, Agonist of MC 3 receptor, CAS No.72629-65-3(free), Agonist of MC 3 receptor

CAS: 72629-65-3(free) Cat. No.: M286707 Peso molecular: 1512.74 (free base)

GRADE & PURITY Moligand™, ≥98%

Descripción general

γ1-MSH TFA is a melanocortin MC3 receptor agonist, with a Ki of 34 nM for the rat MC3 receptor. γ1-MSH TFA displays ~40-fold selectivity over MC4 (Ki=1318 nM).

Specifications

Product Name

γ1-MSH TFA, Agonist of MC 3 receptor, CAS No.72629-65-3(free)

Grado

Moligand™

Especificaciones y pureza

Moligand™, ≥98%

Mecanismos bioquímicos y fisiológicos

Endogenous melanocortin MC3receptor agonist (pKi= 7.46) that displays ~ 40-fold selectivity over MC4. Increases the release of extracellular dopamine, which induces grooming and vertical activity (rearing) in rats. Exhibits hypertensive, tachycardic and s

Secuencia

YVMGHFRWDRF-NH2

Tipo de acción

AGONIST

Mecanismo de acción

Agonist of MC 3 receptor

CAS

72629-65-3(free)

Tipo de molécula

Peptide

Almacenamiento y envío

Condiciones de almacenamiento de almacenamiento

Protected from light,Store at -20°C,Argon charged

Enviado en

Ice chest + Ice pads

Objetivos asociados (humanos)

MC3R Tchem Melanocortin receptor 3 (0 Activities)

Discover Target: MC3R

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Información genética

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