AZ8838 - Moligand™, ≥98% , Antagonist of PAR2, CAS No.2100285-41-2, Antagonist of PAR2

CAS: 2100285-41-2 Cat. No.: A607846 Peso molecular: 234.27 PubChem CID: 132117107
Disponible para pedir
GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
 ·  off list, applied to all prices below.
Size
Estado
Price
Qty
1mg
A607846-1mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
279,90US$
5mg
A607846-5mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
759,90US$
10mg
A607846-10mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
1.199,90US$
25mg
A607846-25mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
1.999,90US$
Enter a quantity for the sizes you want to add.
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Why this grade

Moligand™, ≥98% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

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Storage & shipping

Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.

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Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

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Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Descripción general

AZ8838 is a potent, competitive, allosteric, orally active non-peptide small molecule antagonist of PAR2 with a pKi of 6.4 for hPAR2.

Specifications

Especificaciones y pureza
Moligand™, ≥98%
Condiciones de almacenamiento de almacenamiento
Store at -20°C
Enviado en
Ice chest + Ice pads
Este producto requiere envío en cadena de frío. Los servicios terrestres y otros servicios económicos no están disponibles.
Grado
Moligand™
Tipo de acción
ANTAGONIST
Mecanismo de acción
Antagonist of PAR2
Pureza
≥98%
Nombres e identificadores
Sonrisas canónicasCCCC1=C(C=CC(=C1)F)C(C2=NC=CN2)O
IUPAC Name(R)-(4-fluoro-2-propylphenyl)-(1H-imidazol-2-yl)methanol
InChIKeyIDFPQEHZYBXIFO-GFCCVEGCSA-N
INCHI1S/C13H15FN2O/c1-2-3-9-8-10(14)4-5-11(9)12(17)13-15-6-7-16-13/h4-8,12,17H,2-3H2,1H3,(H,15,16)/t12-/m1/s1
PubChem CID 132117107
Peso molecular 234.27

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Estructura 3D
Modelo de Estructura Química Interactiva





Objetivos asociados (humanos)
F2RL1 Tchem Proteinase-activated receptor 2 (3 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
Certificados (CoA, COO, BSE/TSE y tabla de análisis)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Propiedades químicas y físicas
SolubilidadDMSO:200 mg/mL(853.72mM;Need ultrasonic)
Calculadoras de soluciones
Reseñas

Reseñas de cliente

Need help choosing the grade?

Our grade selection guide covers purity, stabilizer status, and application suitability for all variants in our catalog.

View Moligand™ grade guide →

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