Endomorphin 2 TFA - ≥99% , CAS No.1276124-00-5

CAS: 1276124-00-5 Cat. No.: E650113 Peso molecular: 685.69 PubChem CID: 137700452

GRADE & PURITY ≥99%

Storage

Desiccated,Store at -80°C

Shipped In

Dry ice packs + Cold packs

Descripción general

Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor , displays reasonable affinities for kappa 3 binding sites, with K i value between 20 and 30 nM

Form:Solid

IC50& Target:Ki: 20-30 nM (kappa 3 opioid receptor)

Specifications

Especificaciones y pureza

≥99%

Mecanismos bioquímicos y fisiológicos

Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor , displays reasonable affinities for kappa 3 binding sites, with K i value between 20 and 30 nM.

Condiciones de almacenamiento de almacenamiento

Desiccated, Store at -80°C

Enviado en

Dry ice packs + Cold packs

Este producto requiere envío en cadena de frío. Los servicios terrestres y otros servicios económicos no están disponibles.

Tipo de acción

AGONIST

Pureza

≥99%

Nombres e identificadores

• Sonrisas canónicas: C1CC(N(C1)C(=O)C(CC2=CC=C(C=C2)O)N)C(=O)NC(CC3=CC=CC=C3)C(=O)NC(CC4=CC=CC=C4)C(=O)N.C(=O)(C(F)(F)F)O
• IUPAC Name: (2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-N-[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamide;2,2,2-trifluoroacetic acid
• InChIKey: ONJAQAAWBPIPNC-ZLYCMTQRSA-N
• INCHI: 1S/C32H37N5O5.C2HF3O2/c33-25(18-23-13-15-24(38)16-14-23)32(42)37-17-7-12-28(37)31(41)36-27(20-22-10-5-2-6-11-22)30(40)35-26(29(34)39)19-21-8-3-1-4-9-21;3-2(4,5)1(6)7/h1-6,8-11,13-16,25-28,38H,7,12,17-20,33H2,(H2,34,39)(H,35,40)(H,36,41);(H,6,7)/t25-,26-,27-,28-;/m0./s1
• PubChem CID: 137700452
• Peso molecular: 685.69

Propiedades químicas y físicas

• Solubilidad: H2O : 62.5 mg/mL (91.15 mM; Need ultrasonic) DMSO : 6 mg/mL (8.75 mM; Need ultrasonic)