Gabazine - Moligand™ , Antagonist of GABA A receptor α1 subunit;Antagonist of GABA A receptor α2 subunit;Antagonist of GABA A receptor α3 subunit;Antagonist of GABA A receptor α4 subunit;Antagonist of GABA A receptor α5 subunit;Antagonist of GABA A recept, Antagonist of GABA A receptor α1 subunit;Antagonist of GABA A receptor α2 subunit;Antagonist of GABA A receptor α3 subunit;Antagonist of GABA A receptor α4 subunit;Antagonist of GABA A receptor α5 subunit;Antagonist of GABA A receptor α6 subunit
GRADE & PURITYMoligand™?Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools.
Synonyms
6-imino-3-(4-methoxyphenyl)-1(6h)-pyridazinebutanoic acid | FT-0668923 | 4-(6-Imino-3-(4-methoxyphenyl)-1(6H)-pyridazinyl)butanoic acid | HK Formula No. K 7117 | 1(6H)-Pyridazinebutanoic acid, 6-imino-3-(4-methoxyphenyl)- | BPBio1_000771 | 1,6-Dihydro-6-i
Gabazine is a specific GABA receptor antagonist which does not affect GABA-transaminase or glutamate-decarboxylase activitites.
Specifications
Sinónimos
6-imino-3-(4-methoxyphenyl)-1(6h)-pyridazinebutanoic acid | FT-0668923 | 4-(6-Imino-3-(4-methoxyphenyl)-1(6H)-pyridazinyl)butanoic acid | HK Formula No. K 7117 | 1(6H)-Pyridazinebutanoic acid, 6-imino-3-(4-methoxyphenyl)- | BPBio1_000771 | 1, 6-Dihydro-6-i
Especificaciones y pureza
Moligand™
Condiciones de almacenamiento de almacenamiento
Store at -20°C
Enviado en
Ice chest + Ice pads
Este producto requiere envío en cadena de frío. Los servicios terrestres y otros servicios económicos no están disponibles.
Grado
Moligand™
Tipo de acción
ANTAGONIST
Mecanismo de acción
Antagonist of GABA A receptor α1 subunit;Antagonist of GABA A receptor α2 subunit;Antagonist of GABA A receptor α3 subunit;Antagonist of GABA A receptor α4 subunit;Antagonist of GABA A receptor α5 subunit;Antagonist of GABA A receptor α6 subunit
This compound belongs to the class of organic compounds known as phenylpyridazines. These are organic compounds containing a pyridazine ring substituted by a phenyl group.
External Descriptors
methoxybenzene
1. Djoumbou Feunang Y, Eisner R, Knox C, Chepelev L, Hastings J, Owen G, Fahy E, Steinbeck C, Subramanian S, Bolton E, Greiner R, and Wishart DS. ClassyFire: Automated Chemical Classification With A Comprehensive, Computable Taxonomy. Journal of Cheminformatics, 2016, 8:61.
Certificados (CoA, COO, BSE/TSE y tabla de análisis)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Propiedades químicas y físicas
Solubilidad
Soluble in DMSO and Methanol
Punto de fusión (°C)
244-248° C
Peso molecular
287.310 g/mol
XLogP3
1.400
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
5
Rotatable Bond Count
6
Exact Mass
287.127 Da
Monoisotopic Mass
287.127 Da
Topological Polar Surface Area
86.000 Ų
Heavy Atom Count
21
Formal Charge
0
Complexity
451.000
Isotope Atom Count
0
Defined Atom Stereocenter Count
0
Undefined Atom Stereocenter Count
0
Defined Bond Stereocenter Count
0
Undefined Bond Stereocenter Count
0
The total count of all stereochemical bonds
0
Covalently-Bonded Unit Count
1
Calculadoras de soluciones
Molarity Calculator
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Dilution Calculator
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Reconstitution Calculator
Reseñas
Reseñas de cliente
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