Gabexate Mesylate - 10mM in DMSO , CAS No.56974-61-9

CAS: 56974-61-9 Cat. No.: G408437 Peso molecular: 417.48 Número EC: 611-438-2

GRADE & PURITY 10mM in DMSO

Synonyms

4-​[[6-​[(aminoiminomethyl)​amino]​-​1-​oxohexyl]​oxy]​-benzoic acid ethyl ester,methanesulfonate (1:1)

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

Descripción general

Information

Gabexate Mesylate Gabexate Mesylate is a serine protease inhibitor with IC50 of 0.19 μM which is used therapeutically in the treatment of pancreatitis and disseminated intravascular coagulation.
In vitro

In vivo

Cell Data

cell lines：

Concentrations：

Incubation Time：

Powder Purity:≥99%

Specifications

Sinónimos

4-​[[6-​[(aminoiminomethyl)​amino]​-​1-​oxohexyl]​oxy]​-benzoic acid ethyl ester, methanesulfonate (1:1)

Especificaciones y pureza

10mM in DMSO

Mecanismos bioquímicos y fisiológicos

Gabexate Mesylate is a serine protease inhibitor with IC50 of 0.19 μM which is used therapeutically in the treatment of pancreatitis and disseminated intravascular coagulation.

Condiciones de almacenamiento de almacenamiento

Store at -80°C

Enviado en

Dry ice packs + Cold packs

Este producto requiere envío en cadena de frío. Los servicios terrestres y otros servicios económicos no están disponibles.

Nombres e identificadores

• Isómeros SMILES: CCOC(=O)C1=CC=C(C=C1)OC(=O)CCCCCN=C(N)N.CS(=O)(=O)O
• Peso molecular: 417.48
• Reaxy-Rn: 26001927
• Reaxys-RN_link_address: https://www.reaxys.com/reaxys/secured/hopinto.do?context=S&query=IDE.XRN=26001927&ln=

Propiedades químicas y físicas

• Solubilidad: Solubility (25°C) In vitro DMSO: 100 mg/mL (125.79 mM)
• Punto de fusión (°C): 91 °C

Referencias

1. Wen Zhang, Xu-Dong Wang, Xiao-Han Zhang, Rui Feng, Jun-Long Wang, Wei-Bao Kong, Ji Zhang, Jun-Yu Liang.  (2023)  Biological activities of Elsholtzia stauntoni essential oil and its major constituents against Tribolium castaneum larvae and Lasioderma serricorne adults.  Journal of Essential Oil Bearing Plants,      [PMID:] [10.1080/0972060X.2023.2273262]

2. Han Liu, Yezhou Ni, Jing Hu, Yameng Jin, Peng Gu, Hua Qiu, Kunlin Chen.  (2022)  Self-Healing and Antibacterial Essential Oil-Loaded Mesoporous Silica/Polyacrylate Hybrid Hydrogel for High-Performance Wearable Body-Strain Sensing.  ACS Applied Materials & Interfaces,      [PMID:35500100] [10.1021/acsami.2c03406]