10mM in DMSO for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
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Storage & shipping
Store at -80°C Ships Dry ice packs + Cold packs Check lot-specific COA for exact specifications.
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Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
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Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Descripción general
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC 50 of 19 nM.
In Vitro
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC 50 of 19 nM. MCE has not independently confirmed the accuracy of these methods. They are for reference only.
In Vivo
H4 Receptor antagonist 1 indicates that metabolic stability in rat microsomes is very low with only 1% parent compound remaining after 10 min incubation . MCE has not independently confirmed the accuracy of these methods. They are for reference only.
IC50& Target:H 4 receptor 19 nM (IC 50 )
Specifications
Especificaciones y pureza
10mM in DMSO
Mecanismos bioquímicos y fisiológicos
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC 50 of 19 nM.
Condiciones de almacenamiento de almacenamiento
Store at -80°C
Enviado en
Dry ice packs + Cold packs
Este producto requiere envío en cadena de frío. Los servicios terrestres y otros servicios económicos no están disponibles.
Tipo de acción
INHIBITOR
Nombres e identificadores
Peso molecular
316.79
Documentation
📋 Safety Data Sheet (SDS)
Comprehensive hazard, handling, storage, and regulatory compliance document.
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