LPA2 antagonist 1 - Moligand™,10mM in DMSO , CAS No.1017606-66-4

CAS: 1017606-66-4 Cat. No.: L656453 Peso molecular: 500.46
Disponible para pedir
GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. 10mM in DMSO
Storage
Store at -80°C
Shipped In
Dry ice packs + Cold packs
 ·  off list, applied to all prices below.
Size
Estado
Price
Qty
1ml
L656453-1ml
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
289,90US$
1mg
L656453-1mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
109,90US$
25mg
L656453-25mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
749,90US$
100mg
L656453-100mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
1.469,90US$
250mg
L656453-250mg
8-12 wks(?) Production requires sourcing of materials. We appreciate your patience and understanding.
2.569,90US$
Enter a quantity for the sizes you want to add.
🧪

Why this grade

Moligand™,10mM in DMSO Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

🌡

Storage & shipping

Store at -80°C Ships Dry ice packs + Cold packs Check lot-specific COA for exact specifications.

📋

Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

📚

Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Descripción general

LPA2 antagonist 1 is a LPA2 antagonist with an IC 50 of 17 nM.

In Vitro

LPA2 antagonist 1 inhibits the phosphorylation of Erk induced by LPA in a concentration dependent manner. LPA2 antagonist 1 inhibits HCT-116 colon cancer cell proliferation caused by LPA in a doses dependent manner. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

IC50& Target:IC50: 17 nM (LPA2)

Specifications

Especificaciones y pureza
Moligand™, 10mM in DMSO
Mecanismos bioquímicos y fisiológicos
LPA2 antagonist 1 is a LPA2 antagonist with an IC 50 of 17 nM.
Condiciones de almacenamiento de almacenamiento
Store at -80°C
Enviado en
Dry ice packs + Cold packs
Este producto requiere envío en cadena de frío. Los servicios terrestres y otros servicios económicos no están disponibles.
Grado
Moligand™
Tipo de acción
INHIBITOR
Nombres e identificadores
Isómeros SMILES CC1=CSC2=C1N=CN=C2N[C@@H](C)CN3CCN(CC3)S(=O)(=O)C4=CC(=C(C=C4)Cl)Cl
Peso molecular 500.46

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Objetivos asociados (humanos)
LPAR2 Tchem Lysophosphatidic acid receptor 2 (1 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
Certificados (CoA, COO, BSE/TSE y tabla de análisis)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Calculadoras de soluciones
Reseñas

Reseñas de cliente

Need help choosing the grade?

Our grade selection guide covers purity, stabilizer status, and application suitability for all variants in our catalog.

View Moligand™ grade guide →

Shall we send you a message when we have discounts available?

Remind me later

Thank you! Please check your email inbox to confirm.

Oops! Notifications are disabled.