DCLX069 - ≥98% , CAS No.792946-69-1

CAS: 792946-69-1 Cat. No.: D650930 분자식: C₂₀H₂₅N₃O₂ 분자량: 339.43

GRADE & PURITY ≥98%

Storage

Protected from light,Store at -80°C

Shipped In

Dry ice packs + Cold packs

개요

DCLX069 is a selective protein arginine methyltransferase 1 (PRMT1) inhibitor with an IC 50 value of 17.9 µM. DCLX069 shows less active against PRMT4 and PRMT6 . DCLX069 has anticancer effects

In Vitro

DCLX069 (12.5-100 µM) effectively blocks cell proliferation in breast cancer, liver cancer and acute myeloid leukemia cell lines (MCF7, HepG2, and THP1 cells) in a concentration-dependent manner. MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Form:Solid

IC50& Target:PRMT1 17.9 μM (IC 50 )

Specifications

사양 및 순도

≥98%

생화학 및 생리적 메커니즘

DCLX069 is a selective protein arginine methyltransferase 1 (PRMT1) inhibitor with an IC 50 value of 17.9 µM. DCLX069 shows less active against PRMT4 and PRMT6 . DCLX069 has anticancer effects.

보관 조건

Protected from light,Store at -80°C

배송

Dry ice packs + Cold packs

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작업 유형

INHIBITOR

순수함

≥98%

이름과 식별자

• 분자량: 339.43

화학 및 물리적 특성

• 용해성: DMSO : 100 mg/mL (294.61 mM; Need ultrasonic)