EZM0414 TFA - ≥99% , CAS No.2411759-92-5

CAS: 2411759-92-5 Cat. No.: E651886 분자식: C₂₄H₃₀F₄N₄O₄ 분자량: 514.51 PubChem CID: 155971202

GRADE & PURITY ≥99%

Storage

Store at 2-8°C,Desiccated

Shipped In

Wet ice

개요

EZM0414 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase . EZM0414 TFA has anti-proliferative effects

Form:Solid

IC50& Target:SETD2

Specifications

사양 및 순도

≥99%

생화학 및 생리적 메커니즘

EZM0414 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase . EZM0414 TFA has anti-proliferative effects.

보관 조건

Store at 2-8°C,Desiccated

배송

Wet ice

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작업 유형

INHIBITOR

순수함

≥99%

이름과 식별자

• 정식 스마일: CC1=C2C(=C(C=C1)F)C=C(N2)C(=O)NC3CCCC(C3)N4CCN(CC4)C(=O)C.C(=O)(C(F)(F)F)O
• IUPAC Name: N-[(1R,3S)-3-(4-acetylpiperazin-1-yl)cyclohexyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide;2,2,2-trifluoroacetic acid
• InChIKey: HASNOYOGMISGTP-PPPUBMIESA-N
• INCHI: 1S/C22H29FN4O2.C2HF3O2/c1-14-6-7-19(23)18-13-20(25-21(14)18)22(29)24-16-4-3-5-17(12-16)27-10-8-26(9-11-27)15(2)28;3-2(4,5)1(6)7/h6-7,13,16-17,25H,3-5,8-12H2,1-2H3,(H,24,29);(H,6,7)/t16-,17+;/m1./s1
• PubChem CID: 155971202
• 분자량: 514.51

화학 및 물리적 특성

• 용해성: DMSO : 200 mg/mL (388.72 mM; Need ultrasonic) H2O : 6.67 mg/mL (12.96 mM; ultrasonic and warming and heat to 60°C)