PROTAC ERRα ligand 2 - 10mM in DMSO , CAS No.2306388-57-6

CAS: 2306388-57-6 Cat. No.: P655477 분자식: C₂₀H₁₃F₆NO₄ 분자량: 445.3 PubChem CID: 139291005

GRADE & PURITY 10mM in DMSO

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

개요

PROTAC ERRα ligand 2 is an estrogen-related receptor α ( ERRα ) inverse agonist with an IC 50 of 5.67 nM. PROTAC ERRα ligand 2 (IC 50 =5.67 nM) displays a ~11-fold improved potency than XCT790 (IC 50 =61.3 nM).

Specifications

사양 및 순도

10mM in DMSO

생화학 및 생리적 메커니즘

PROTAC ERRα ligand 2 is an estrogen-related receptor α ( ERRα ) inverse agonist with an IC 50 of 5.67 nM. PROTAC ERRα ligand 2 (IC 50 =5.67 nM) displays a ~11-fold improved potency than XCT790 (IC 50 =61.3 nM).

보관 조건

Store at -80°C

배송

Dry ice packs + Cold packs

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작업 유형

ANTAGONIST

이름과 식별자

• 이성체 SMILES: COC1=C(C=CC(=C1)/C=C(\C#N)/C(=O)O)OCC2=C(C=C(C=C2)C(F)(F)F)C(F)(F)F
• PubChem CID: 139291005
• 분자량: 445.3

관련 대상(인간)

ESRRA Tchem Steroid hormone receptor ERR1 (1 Activities)

Discover Target: ESRRA

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

자주 묻는 질문

How should this product be stored?

Store at ?80 °C. Ultra-low temperature storage is required to maintain the specified shelf life.

How is this product shipped?

This product ships frozen with dry ice and cold packs. Unpack on arrival and transfer it to the storage condition stated above; handle dry ice with insulated gloves in a ventilated area.

What are the CAS number, molecular formula and molecular weight?

The CAS Number is 2306388-57-6, the molecular formula is C20H13F6NO4, and the molecular weight is 445.3 g/mol.

What documentation is provided?

Available product documentation, including Certificates of Analysis (COA), Safety Data Sheets (SDS), and specification sheets, is shown in the product document area. Document availability and access follow the current site policy.