Rebamipide - Moligand™, 10mM in DMSO , Agonist of CCK 1 receptor, CAS No.90098-04-7, Agonist of CCK 1 receptor

CAS: 90098-04-7 Cat. No.: R408057 분자식: C₁₉H₁₅ClN₂O₄.xH₂O 분자량: 370.79 EC 번호: 815-380-0 PubChem CID: 5042

GRADE & PURITY Moligand™, 10mM in DMSO

Synonyms

OPC-12759 | α-​[(4-​chlorobenzoyl)​amino]​-​1,​2-​dihydro-​2-​oxo-4-​quinolinepropanoic acid

Storage

Store at -80°C

Shipped In

Dry ice packs + Cold packs

개요

Information

Rebamipide Rebamipide (OPC-12759) is a cholecystokinin type 1 (CCK1) receptor inhibitor for inhibiting [ 125 I]BH-CCK-8S with IC50 of 37.7 μM.
In vitro

In vivo

Cell Data

cell lines：

Concentrations：

Incubation Time：

Powder Purity:≥99%

Specifications

동의어

OPC-12759 | α-​[(4-​chlorobenzoyl)​amino]​-​1,​2-​dihydro-​2-​oxo-4-​quinolinepropanoic acid

사양 및 순도

Moligand™, 10mM in DMSO

생화학 및 생리적 메커니즘

Rebamipide (OPC-12759) is a cholecystokinin type 1 (CCK1) receptor inhibitor for inhibiting [¹²⁵I]BH-CCK-8S with IC50 of 37.7 μM.

보관 조건

Store at -80°C

배송

Dry ice packs + Cold packs

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등급

Moligand™

작업 유형

AGONIST

작동 메커니즘

Agonist of CCK 1 receptor

이름과 식별자

• 이성체 SMILES: C1=CC=C2C(=C1)C(=CC(=O)N2)CC(C(=O)O)NC(=O)C3=CC=C(C=C3)Cl
• RTECS: VC2518500
• PubChem CID: 5042
• 분자량: 370.79
• Reaxy-Rn: 5384689

관련 대상(인간)

CCKAR Tclin Cholecystokinin receptor type A (1 Activities)

Discover Target: CCKAR

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

화학 및 물리적 특성

• 녹는점(°C): 290°C(dec.)(lit.)

참고 문헌

1. Han Qiao, Zhuo Xu, Mengchi Sun, Shuwen Fu, Fangxue Zhao, Danping Wang, Zhonggui He, Yinglei Zhai, Jin Sun.  (2022)  Rebamipide liposome as an effective ocular delivery system for the management of dry eye disease.  JOURNAL OF DRUG DELIVERY SCIENCE AND TECHNOLOGY,      [PMID:] [10.1016/j.jddst.2022.103654]