AC187, Antagonist of AMY 1 receptor;Antagonist of AMY 3 receptor;Antagonist of CT receptor, CAS No.151804-77-2, Antagonist of AMY 1 receptor;Antagonist of AMY 3 receptor;Antagonist of CT receptor

CAS: 151804-77-2 Cat. No.: rp173362 Formule: C₁₂₇H₂₀₅N₃₇O₄₀ Poids moléculaire: 2890.24 PubChem CID: 16133792

GRADE & PURITY Moligand™

Specifications

Product Name

AC187, Antagonist of AMY 1 receptor;Antagonist of AMY 3 receptor;Antagonist of CT receptor, CAS No.151804-77-2

Synonymes

AC 187;AC-187;acetyl-(Asn³⁰,Tyr³²)-calcitonin⁸⁻³²;salmon calcitonin (8-32) reduced

Grade

Moligand™

Spécifications et pureté

Moligand™

Type d'action

ANTAGONIST

Mécanisme d'action

Antagonist of AMY 1 receptor;Antagonist of AMY 3 receptor;Antagonist of CT receptor

CAS

151804-77-2

Type de molécule

Peptide

Stockage et expédition

Conditions de stockage de stockage

Room temperature

Taxonomic Classification

Taxonomy Tree

• Kingdom Organic compounds
  • Superclass Organic Polymers
    • Classe Polypeptides

• Kingdom: Organic compounds
• Superclass: Organic Polymers
• Classe: Polypeptides
• Subclass: Not available
• Intermediate Tree Nodes: Not available
• Direct Parent: Polypeptides
• Alternative Parents: Peptides Tyrosine and derivatives Arginine and derivatives Phenylalanine and derivatives Histidine and derivatives Glutamic acid and derivatives Glutamine and derivatives Asparagine and derivatives Leucine and derivatives Valine and derivatives Proline and derivatives N-acyl-alpha amino acids and derivatives Serine and derivatives Alpha amino acid amides Amphetamines and derivatives Pyrrolidinecarboxamides Imidazolyl carboxylic acids and derivatives N-acylpyrrolidines 1-hydroxy-2-unsubstituted benzenoids N-acyl amines Acetamides Tertiary carboxylic acid amides Heteroaromatic compounds Secondary carboxylic acid amides Primary carboxylic acid amides Guanidines Amino acids Secondary alcohols Monocarboxylic acids and derivatives Carboxylic acids Azacyclic compounds Carboximidamides Hydrocarbon derivatives Imines Organic oxides Primary alcohols Carbonyl compounds Monoalkylamines
• Molecular Framework: Aromatic heteromonocyclic compounds
• Substituents: Polypeptide - Alpha peptide - Tyrosine or derivatives - Arginine or derivatives - Phenylalanine or derivatives - Histidine or derivatives - Glutamic acid or derivatives - Glutamine or derivatives - Asparagine or derivatives - Leucine or derivatives - Valine or derivatives - N-acyl-alpha amino acid or derivatives - Proline or derivatives - Serine or derivatives - Alpha-amino acid amide - Alpha-amino acid or derivatives - N-substituted-alpha-amino acid - Amphetamine or derivatives - N-acylpyrrolidine - Pyrrolidine carboxylic acid or derivatives - Pyrrolidine-2-carboxamide - Imidazolyl carboxylic acid derivative - Phenol - 1-hydroxy-2-unsubstituted benzenoid - Benzenoid - N-acyl-amine - Fatty amide - Fatty acyl - Monocyclic benzene moiety - Heteroaromatic compound - Imidazole - Tertiary carboxylic acid amide - Azole - Pyrrolidine - Acetamide - Amino acid or derivatives - Amino acid - Carboxamide group - Guanidine - Secondary carboxylic acid amide - Secondary alcohol - Primary carboxylic acid amide - Monocarboxylic acid or derivatives - Azacycle - Carboxylic acid derivative - Carboximidamide - Carboxylic acid - Organoheterocyclic compound - Primary alcohol - Organic oxide - Amine - Organic oxygen compound - Carbonyl group - Imine - Hydrocarbon derivative - Primary aliphatic amine - Alcohol - Organic nitrogen compound - Primary amine - Organonitrogen compound - Organooxygen compound - Aromatic heteromonocyclic compound
• Description: This compound belongs to the class of organic compounds known as polypeptides. These are peptides containing ten or more amino acid residues.
• External Descriptors: Not available

Data sources

1. Djoumbou Feunang Y, Eisner R, Knox C, Chepelev L, Hastings J, Owen G, Fahy E, Steinbeck C, Subramanian S, Bolton E, Greiner R, and Wishart DS. ClassyFire: Automated Chemical Classification With A Comprehensive, Computable Taxonomy. Journal of Cheminformatics, 2016, 8:61.

DOI: 10.1186/s13321-016-0174-y

Cibles associées (humaines)

RAMP1 Tclin Receptor activity-modifying protein 1 (0 Activities)

Discover Target: RAMP1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

RAMP3 Tclin Receptor activity-modifying protein 3 (0 Activities)

Discover Target: RAMP3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

CALCR Tclin Calcitonin receptor (0 Activities)

Discover Target: CALCR

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Informations génétiques

• Alternate Names: AC 187;AC-187;acetyl-(Asn³⁰,Tyr³²)-calcitonin⁸⁻³²;salmon calcitonin (8-32) reduced
• Reference:
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Foire aux questions

What is Moligand??

Moligand? is one of Aladdin Scientific's premium product lines, formulated for high-purity applications across multiple workflows. Compared to standard grades in the same workflow, Moligand? products typically offer tighter specifications, more rigorous QC, and stronger lot-to-lot consistency.

How should this product be stored?

Store at room temperature.

What are the CAS number, molecular formula and molecular weight?

The CAS Number is 151804-77-2. InChIKey ZLFXHYNEZYAYPG-AABHONRUSA-N.

What documentation is provided?

Available product documentation, including Certificates of Analysis (COA), Safety Data Sheets (SDS), and specification sheets, is shown in the product document area. Document availability and access follow the current site policy.