AC187, Antagonist of AMY 1 receptor;Antagonist of AMY 3 receptor;Antagonist of CT receptor, CAS No.151804-77-2, Antagonist of AMY 1 receptor;Antagonist of AMY 3 receptor;Antagonist of CT receptor

CAS: 151804-77-2 Cat. No.: rp173362 Molecular Weight: 2890.24 PubChem CID: 16133792

GRADE & PURITY Moligand™

Specifications

Product Name

AC187, Antagonist of AMY 1 receptor;Antagonist of AMY 3 receptor;Antagonist of CT receptor, CAS No.151804-77-2

Synonyms

AC 187;AC-187;acetyl-(Asn³⁰, Tyr³²)-calcitonin⁸⁻³²;salmon calcitonin (8-32) reduced

Grade

Moligand™

Specifications & Purity

Moligand™

Action Type

ANTAGONIST

Mechanism of action

Antagonist of AMY 1 receptor;Antagonist of AMY 3 receptor;Antagonist of CT receptor

CAS

151804-77-2

Molecule Type

Peptide

Storage and Shipping

Storage

Room temperature

Taxonomic Classification

Taxonomy Tree

• Kingdom Organic compounds
  • Superclass Organic Polymers
    • Class Polypeptides

• Kingdom: Organic compounds
• Superclass: Organic Polymers
• Class: Polypeptides
• Subclass: Not available
• Intermediate Tree Nodes: Not available
• Direct Parent: Polypeptides
• Alternative Parents: Peptides Tyrosine and derivatives Arginine and derivatives Phenylalanine and derivatives Histidine and derivatives Glutamic acid and derivatives Glutamine and derivatives Asparagine and derivatives Leucine and derivatives Valine and derivatives Proline and derivatives N-acyl-alpha amino acids and derivatives Serine and derivatives Alpha amino acid amides Amphetamines and derivatives Pyrrolidinecarboxamides Imidazolyl carboxylic acids and derivatives N-acylpyrrolidines 1-hydroxy-2-unsubstituted benzenoids N-acyl amines Acetamides Tertiary carboxylic acid amides Heteroaromatic compounds Secondary carboxylic acid amides Primary carboxylic acid amides Guanidines Amino acids Secondary alcohols Monocarboxylic acids and derivatives Carboxylic acids Azacyclic compounds Carboximidamides Hydrocarbon derivatives Imines Organic oxides Primary alcohols Carbonyl compounds Monoalkylamines
• Molecular Framework: Aromatic heteromonocyclic compounds
• Substituents: Polypeptide - Alpha peptide - Tyrosine or derivatives - Arginine or derivatives - Phenylalanine or derivatives - Histidine or derivatives - Glutamic acid or derivatives - Glutamine or derivatives - Asparagine or derivatives - Leucine or derivatives - Valine or derivatives - N-acyl-alpha amino acid or derivatives - Proline or derivatives - Serine or derivatives - Alpha-amino acid amide - Alpha-amino acid or derivatives - N-substituted-alpha-amino acid - Amphetamine or derivatives - N-acylpyrrolidine - Pyrrolidine carboxylic acid or derivatives - Pyrrolidine-2-carboxamide - Imidazolyl carboxylic acid derivative - Phenol - 1-hydroxy-2-unsubstituted benzenoid - Benzenoid - N-acyl-amine - Fatty amide - Fatty acyl - Monocyclic benzene moiety - Heteroaromatic compound - Imidazole - Tertiary carboxylic acid amide - Azole - Pyrrolidine - Acetamide - Amino acid or derivatives - Amino acid - Carboxamide group - Guanidine - Secondary carboxylic acid amide - Secondary alcohol - Primary carboxylic acid amide - Monocarboxylic acid or derivatives - Azacycle - Carboxylic acid derivative - Carboximidamide - Carboxylic acid - Organoheterocyclic compound - Primary alcohol - Organic oxide - Amine - Organic oxygen compound - Carbonyl group - Imine - Hydrocarbon derivative - Primary aliphatic amine - Alcohol - Organic nitrogen compound - Primary amine - Organonitrogen compound - Organooxygen compound - Aromatic heteromonocyclic compound
• Description: This compound belongs to the class of organic compounds known as polypeptides. These are peptides containing ten or more amino acid residues.
• External Descriptors: Not available

Data sources

1. Djoumbou Feunang Y, Eisner R, Knox C, Chepelev L, Hastings J, Owen G, Fahy E, Steinbeck C, Subramanian S, Bolton E, Greiner R, and Wishart DS. ClassyFire: Automated Chemical Classification With A Comprehensive, Computable Taxonomy. Journal of Cheminformatics, 2016, 8:61.

DOI: 10.1186/s13321-016-0174-y

Associated Targets(Human)

RAMP1 Tclin Receptor activity-modifying protein 1 (0 Activities)

Discover Target: RAMP1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

RAMP3 Tclin Receptor activity-modifying protein 3 (0 Activities)

Discover Target: RAMP3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

CALCR Tclin Calcitonin receptor (0 Activities)

Discover Target: CALCR

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)

Genetic information

• Alternate Names: AC 187;AC-187;acetyl-(Asn³⁰,Tyr³²)-calcitonin⁸⁻³²;salmon calcitonin (8-32) reduced
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