AZ8838 - Moligand™, ≥98% , Antagonist of PAR2, CAS No.2100285-41-2, Antagonist of PAR2

CAS: 2100285-41-2 Cat. No.: A607846 Formule: C13H15FN2O Poids moléculaire: 234.27 PubChem CID: 132117107
DISPONIBLE À COMMANDE
GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
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Size
Allemagne (EU)
USA*
Price
Qty
1mg
A607846-1mg
Sur commande · 8–12 semaines
242,88€
5mg
A607846-5mg
Sur commande · 8–12 semaines
659,39€
10mg
A607846-10mg
Sur commande · 8–12 semaines
1 041,20€
25mg
A607846-25mg
Sur commande · 8–12 semaines
1 735,39€
Enter a quantity for the sizes you want to add.
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Why this grade

Moligand™, ≥98% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

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Storage & shipping

Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.

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Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

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Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Vue d’ensemble

AZ8838 is a potent, competitive, allosteric, orally active non-peptide small molecule antagonist of PAR2 with a pKi of 6.4 for hPAR2.

Specifications

Spécifications et pureté
Moligand™, ≥98%
Conditions de stockage de stockage
Store at -20°C
Expédié en
Ice chest + Ice pads
Ce produit nécessite l'expédition en chaîne froide. Les services terrestres et autres services économiques ne sont pas disponibles.
Grade
Moligand™
Type d'action
ANTAGONIST
Mécanisme d'action
Antagonist of PAR2
Pureté
≥98%
Noms et identifiants
Sourires canoniquesCCCC1=C(C=CC(=C1)F)C(C2=NC=CN2)O
IUPAC Name(R)-(4-fluoro-2-propylphenyl)-(1H-imidazol-2-yl)methanol
InChIKeyIDFPQEHZYBXIFO-GFCCVEGCSA-N
INCHI1S/C13H15FN2O/c1-2-3-9-8-10(14)4-5-11(9)12(17)13-15-6-7-16-13/h4-8,12,17H,2-3H2,1H3,(H,15,16)/t12-/m1/s1
PubChem CID 132117107
Poids moléculaire 234.27

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

Structure 3D
Modèle de structure chimique interactif





Cibles associées (humaines)
F2RL1 Tchem Proteinase-activated receptor 2 (3 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
Certificats (CoA, COO, BSE/TSE et tableau d'analyse)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Propriétés chimiques et physiques
SolubilitéDMSO:200 mg/mL(853.72mM;Need ultrasonic)
Calculateurs de solution
Avis

Avis des clients

Need help choosing the grade?

Our grade selection guide covers purity, stabilizer status, and application suitability for all variants in our catalog.

View Moligand™ grade guide →

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