TL12-186 - Moligand™, 10 mM in DMSO , CAS No.2250025-88-6
En stock
SKU
T1496053
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TL12-186 is a Cereblon -dependent multi-kinase PROTAC degrader. Multi-kinases include CDK , BTK , FLT3 , Aurora kinases , TEC , ULK , ITK , et al. TL12-186 inhibits CDK2/cyclin A ( IC 50 =73 nM) and CDK9/cyclin T1 ( IC 50 =55 nM).
| CAS | 2250025-88-6 |
|---|---|
| Concentration | 10 mM in DMSO |
| Spécifications et pureté | Moligand™, 10 mM in DMSO |
| Conditions de stockage de stockage | Protected from light,Desiccated,Store at -80°C |
| Expédié en | Dry ice packs + Cold packs |
| Product Description | TL12-186 is a Cereblon -dependent multi-kinase PROTAC degrader. Multi-kinases include CDK , BTK , FLT3 , Aurora kinases , TEC , ULK , ITK , et al. TL12-186 inhibits CDK2/cyclin A ( IC 50 =73 nM) and CDK9/cyclin T1 ( IC 50 =55 nM). |