PERK
상품
- GSK PERK inhibitor, Inhibitor of eukaryotic translation initiation factor 2 alpha kinase 3;Inhibitor of myosin light chain kinase 2CAS: 1337531-89-1 분자식: C24H19F4N5O 분자량: 469.43Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%● 재고 있음 — 미국 항목 #: G355474상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- 1-[5-(4-amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydroindol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanone
- SMILES
- CN1C=C(C2=C(N=CN=C21)N)C3=CC4=C(C=C3)N(CC4)C(=O)CC5=CC(=CC(=C5)F)C(F)(F)F
- InChIKey
- PXVQGBJMIQCDEX-UHFFFAOYSA-N
- InChI
- show more
- Synonyms
- 1-[5-(4-amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-2, 3-dihydroindol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]eth...
- GSK2606414CAS: 1337531-36-8 분자식: C24H20F3N5O 분자량: 451.44Solid Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%● 재고 있음 — 미국 항목 #: G125654상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- 1-[5-(4-amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydroindol-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanone
- SMILES
- CN1C=C(C2=C(N=CN=C21)N)C3=CC4=C(C=C3)N(CC4)C(=O)CC5=CC(=CC=C5)C(F)(F)F
- InChIKey
- SIXVRXARNAVBTC-UHFFFAOYSA-N
- InChI
- show more
- Synonyms
- AC-29016 | 1-(5-(4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)indolin-1-yl)-2-(3-(trifluoromethyl)phenyl)ethanone...
- GSK2656157, Inhibitor of eukaryotic translation initiation factor 2 alpha kinase 3CAS: 1337532-29-2 분자식: C23H21FN6O 분자량: 416.45Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%● 재고 있음 — 미국 항목 #: G276179상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- 1-[5-(4-amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydroindol-1-yl]-2-(6-methylpyridin-2-yl)ethanone
- SMILES
- CC1=NC(=CC=C1)CC(=O)N2CCC3=C2C=CC(=C3F)C4=CN(C5=NC=NC(=C45)N)C
- InChIKey
- PRWSIEBRGXYXAJ-UHFFFAOYSA-N
- InChI
- show more
- Synonyms
- 1-[5-(4-Amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydro-1H-indol-1-yl]-2-(6-methyl-2-pyridinyl)e...
- ONO 8130, Antagonist of EP 1 receptorCAS: 459841-96-4 분자식: C25H28N2O5S2 분자량: 500.63Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%(HPLC)◐ .주문제작 · 8~12주 항목 #: O287851상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- 4-[[6-[2-methylpropyl-[(4-methyl-1,3-thiazol-2-yl)sulfonyl]amino]-2,3-dihydro-1H-inden-5-yl]oxymethyl]benzoic acid
- SMILES
- CC1=CSC(=N1)S(=O)(=O)N(CC(C)C)C2=C(C=C3CCCC3=C2)OCC4=CC=C(C=C4)C(=O)O
- InChIKey
- IOXMDBQCUCDLAF-UHFFFAOYSA-N
- InChI
- show more
- Synonyms
- AC-36636 | BDBM190564 | 4-[[6-[2-methylpropyl-[(4-methyl-1,3-thiazol-2-yl)sulfonyl]amino]-2,3-dihydro-1H-inden-5-yl]o...
- VU 0424465, Agonist of mGlu 5 receptor;Allosteric modulator of mGlu 5 receptorMoligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%(HPLC)◐ .주문제작 · 8~12주 항목 #: V286883상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- 5-[2-(3-fluorophenyl)ethynyl]-N-[(2R)-3-hydroxy-3-methylbutan-2-yl]pyridine-2-carboxamide
- SMILES
- CC(C(C)(C)O)NC(=O)C1=NC=C(C=C1)C#CC2=CC(=CC=C2)F
- InChIKey
- ZPKZAFDYFVJULO-CYBMUJFWSA-N
- InChI
- 1S/C19H19FN2O2/c1-13(19(2,3)24)22-18(23)17-10-9-15(12-21-17)8-7-14-5-4-6-16(20)11-14/h4-6,9-13,24H,1-3H3,(H,22,23)/t13-/m1/s1
- Synonyms
- 5-[2-(2-(3-Fluorophenyl)ethynyl]-N-[(1R)-2-hydroxy-1,2-dimethylpropyl]-2-pyridinecarboxamide
- AMG PERK 44CAS: 1883548-84-2 분자식: C34H28N4O2•HCl 분자량: 561.07● 재고 있음 — 미국 항목 #: A286749상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- 4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenylpyrazol-3-one;hydrochloride
- SMILES
- CC1=C(C(=C(C=C1)C(=O)C2=C(N(N(C2=O)C3=CC=CC=C3)C)C4=CC=CC=C4)N)C5=CC6=C(C=C5)N=C(C=C6)C.Cl
- InChIKey
- RNAKBTDDCHJCMT-UHFFFAOYSA-N
- InChI
- show more
- Synonyms
- 4-[2-Amino-4-methyl-3-(2-methyl-6-quinolinyl)benzoyl]-1,2-dihydro-1-methyl-2,5-diphenyl-3H-pyrazol-3-one hydrochloride
- NSC 295642CAS: 77111-29-6 분자식: C15H14ClCuN3S2 분자량: 399.42◐ .주문제작 · 8~12주 항목 #: N352361상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- (E)-benzylsulfanyl-[(E)-1-pyridin-2-ylethylidenehydrazinylidene]-sulfidomethane;chlorocopper(1+)
- SMILES
- CC(=NN=C([S-])SCC1=CC=CC=C1)C2=CC=CC=N2.Cl[Cu+]
- InChIKey
- MGXCRQNCPJBYKM-CWQUOYFRSA-L
- InChI
- 1S/C15H15N3S2.ClH.Cu/c1-12(14-9-5-6-10-16-14)17-18-15(19)20-11-13-7-3-2-4-8-13;;/h2-10H,11H2,1H3,(H,18,19);1H;/q;;+2/p-2/b17-12+;;
- Synonyms
- (E)-벤질설파닐-[(E)-1-피리딘-2-에틸리덴하이드라지닐리덴]-설피도메탄;클로로구리(1+) | DTXSID20444568 | NSC 295642 | NSC295642
- ISRIB(트랜스 이성질체)CAS: 1597403-47-8 분자식: C22H24Cl2N2O4 분자량: 451.34● 재고 있음 — 미국 항목 #: I275318상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- 2-(4-chlorophenoxy)-N-[4-[[2-(4-chlorophenoxy)acetyl]amino]cyclohexyl]acetamide
- SMILES
- C1CC(CCC1NC(=O)COC2=CC=C(C=C2)Cl)NC(=O)COC3=CC=C(C=C3)Cl
- InChIKey
- HJGMCDHQPXTGAV-UHFFFAOYSA-N
- InChI
- show more
- Synonyms
- ISRIB | ISRIB trans-isomer | BCP23947 | ISRIB, >=98% (HPLC) | N,N'-(Cyclohexane-1,4-diyl)bis(2-(4-chlorophenoxy)aceta...
- S-(Carboxymethyl)-L-cysteine● 재고 있음 — 미국 항목 #: S161422상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- (2R)-2-amino-3-(carboxymethylsulfanyl)propanoic acid
- SMILES
- N[C@@H](CSCC(O)=O)C(O)=O
- InChIKey
- GBFLZEXEOZUWRN-VKHMYHEASA-N
- InChI
- 1S/C5H9NO4S/c6-3(5(9)10)1-11-2-4(7)8/h3H,1-2,6H2,(H,7,8)(H,9,10)/t3-/m0/s1
- Synonyms
- Carbocysteine, L Isomer | Chilvax | Mucodyne | (2R)-2-amino-3-(carboxymethylsulfanyl)propanoic acid | (2R)-2-amino-3-...
- GSK2656157, Inhibitor of eukaryotic translation initiation factor 2 alpha kinase 3CAS: 1337532-29-2 분자식: C23H21FN6O 분자량: 416.45Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. 10mM in DMSO● 재고 있음 — 미국 항목 #: G421276상품 보기가격 및 팩 크기
기술적 식별자
- IUPAC 이름
- 1-[5-(4-amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydroindol-1-yl]-2-(6-methylpyridin-2-yl)ethanone
- SMILES
- CC1=NC(=CC=C1)CC(=O)N2CCC3=C2C=CC(=C3F)C4=CN(C5=NC=NC(=C45)N)C
- InChIKey
- PRWSIEBRGXYXAJ-UHFFFAOYSA-N
- InChI
- show more
- Synonyms
- 1-[5-(4-Amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydro-1H-indol-1-yl]-2-(6-methyl-2-pyridinyl)e...
빠른 배송 주식 상품에 대한 같은 날 배송
기술적 세부사항 모든 제품 페이지의 품질 및 사양 정보
팩 크기 옵션 목록에서 가격 액세스를 가진 여러 포장 크기
연구 및 개발용 연구 개발용 제품
자주 묻는 질문
How is the PERK listing put together?
It draws on reported PERK annotations within Cell Cycle/DNA Damage and lists each compound with its structure, identifiers, and the activity published for it. Always check the underlying assay before comparing potency values across entries.
How do I choose a PERK modulator for my assay?
Start from the assay format and readout — biochemical, cell-based, or in vivo — then compare the PERK entries on potency, selectivity over related family members, and solubility in your vehicle. Where several chemotypes are available, a reference compound plus a structurally unrelated backup is the usual way to control for off-target effects.
Which specifications matter most for PERK compounds?
Purity and identity confirmation come first, then solubility in DMSO or your chosen vehicle, recommended storage temperature, and stability in solution. For PERK work in particular, freshly prepared stocks avoid most of the reproducibility problems seen with stored plates. All products are supplied for professional research and development use only, and are not for use in humans, animals, diagnostics, or therapy.
What if the PERK compound I need is not listed?
Search by CAS number or SMILES first, since analogs of PERK compounds are often catalogued under a related target. Custom synthesis and bulk enquiries go to [email protected]. We supply verified businesses, research institutions, universities, and government agencies.