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Angiopeptin TFA - ≥99% , CAS No.2478421-60-0
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GRADE & PURITY ≥99%
Storage
Desiccated,Store at -80°C
Shipped In
Dry ice packs + Cold packs
🌎 Ship to: United States
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Why this grade
≥99% for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
Storage & shipping
Desiccated,Store at -80°C Ships Dry ice packs + Cold packs Check lot-specific COA for exact specifications.
Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Übersicht
Angiopeptin TFA, a cyclic octapeptide analogue of somatostatin, is a weak sst 2 /sst 5 receptor partial agonist with IC 50 values of 0.26 nM and 6.92 nM, respectively. Angiopeptin TFA is a potent inhibitor of growth hormone release and insulin-like growth factor-1 (IGF-1) production. Angiopeptin TFA inhibits adenylate cyclase or stimulates extracellular acidification. Angiopeptin TFA has the potential for coronary atherosclerosis research
In Vitro
Angiopeptin (0.1 nM- 10 μM; for 1 h) TFA acts as a partial agonist (pEC 50 =6.57) with a maximum response of 423% at 3 μM on the release of tritium on CHO hsst 2 cells. MCE has not independently confirmed the accuracy of these methods. They are for reference only.
In Vivo
Angiopeptin (20 and 50μg/kg; i.h.) TFA significantly inhibits neointimal formation . Angiopeptin (20 μg/kg; per day) TFA significantly inhibits coronary artery myointimal proliferation in cardiac allografts by appmximalely 50% . MCE has not independently confirmed the accuracy of these methods. They are for reference only.
Form:Solid
IC50& Target:IC50: 0.26 nM (sst2) and 6.92 nM (sst5)
Specifications
Spezifikationen & Reinheit
≥99%
Biochemische und physiologische Mechanismen
Angiopeptin TFA, a cyclic octapeptide analogue of somatostatin, is a weak sst 2 /sst 5 receptor partial agonist with IC 50 values of 0.26u2009nM and 6.92u2009nM, respectively. Angiopeptin TFA is a potent inhibitor of growth hormone release and insulin-lik
Storage
Desiccated,Store at -80°C
Verschickt in
Dry ice packs + Cold packs
Dieses Produkt erfordert Kühlkettenversand. Grundversand und andere Economy-Optionen sind nicht verfügbar.
Aktionsart
AGONIST
Reinheit
≥99%
Namen und Kennungen
| Molekulargewicht | 1326.39 |
|---|
Documentation
📋 Safety Data Sheet (SDS)
Comprehensive hazard, handling, storage, and regulatory compliance document.
Download SDS →✅ Certificate of Analysis (COA)
Lot-specific quality data. Enter your lot number to retrieve the exact COA.
Look up COA →🔬 Specification Sheet
Full quality attributes and acceptance criteria for this grade.
View spec sheet →Advanced Data
Zertifikate (CoA, COO, BSE/TSE und Analyse-Diagramm)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Chemische und physikalische Eigenschaften
| Löslichkeit | H2O : 10 mg/mL (7.54 mM; Need ultrasonic) |
|---|
Lösungsrechner
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