AZ8838 - Moligand™, ≥98% , Antagonist of PAR2, CAS No.2100285-41-2, Antagonist of PAR2

CAS: 2100285-41-2 Cat. No.: A607846 Summenformel: C13H15FN2O Molekulargewicht: 234.27 PubChem CID: 132117107
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GRADE & PURITY Moligand™ ? Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools. ≥98%
Storage
Store at -20°C
Shipped In
Ice chest + Ice pads
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Size
Deutschland (EU)
USA*
Price
Qty
1mg
A607846-1mg
Auf Bestellung · 8–12 Wochen
242,88€
5mg
A607846-5mg
Auf Bestellung · 8–12 Wochen
659,39€
10mg
A607846-10mg
Auf Bestellung · 8–12 Wochen
1.041,20€
25mg
A607846-25mg
Auf Bestellung · 8–12 Wochen
1.735,39€
Enter a quantity for the sizes you want to add.
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Why this grade

Moligand™, ≥98% Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.

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Storage & shipping

Store at -20°C Ships Ice chest + Ice pads Check lot-specific COA for exact specifications.

📋

Quality documents

SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.

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Literature proof

Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.

Übersicht

AZ8838 is a potent, competitive, allosteric, orally active non-peptide small molecule antagonist of PAR2 with a pKi of 6.4 for hPAR2.

Specifications

Spezifikationen & Reinheit
Moligand™, ≥98%
Storage
Store at -20°C
Verschickt in
Ice chest + Ice pads
Dieses Produkt erfordert Kühlkettenversand. Grundversand und andere Economy-Optionen sind nicht verfügbar.
Note
Moligand™
Aktionsart
ANTAGONIST
Mechanismus der Wirkung
Antagonist of PAR2
Reinheit
≥98%
Namen und Kennungen
Kanonisches LächelnCCCC1=C(C=CC(=C1)F)C(C2=NC=CN2)O
IUPAC Name(R)-(4-fluoro-2-propylphenyl)-(1H-imidazol-2-yl)methanol
InChIKeyIDFPQEHZYBXIFO-GFCCVEGCSA-N
INCHI1S/C13H15FN2O/c1-2-3-9-8-10(14)4-5-11(9)12(17)13-15-6-7-16-13/h4-8,12,17H,2-3H2,1H3,(H,15,16)/t12-/m1/s1
PubChem CID 132117107
Molekulargewicht 234.27

Documentation

📋 Safety Data Sheet (SDS)

Comprehensive hazard, handling, storage, and regulatory compliance document.

Download SDS →

✅ Certificate of Analysis (COA)

Lot-specific quality data. Enter your lot number to retrieve the exact COA.

Look up COA →

📊 Datasheet

Quick-reference summary of product specifications and applications.

View datasheet →

🔬 Specification Sheet

Full quality attributes and acceptance criteria for this grade.

View spec sheet →

Advanced Data

3D-Struktur
Interaktives chemisches Strukturmodell





Zugehörige Ziele (menschlich)
F2RL1 Tchem Proteinase-activated receptor 2 (3 Activities)
Activity TypeActivity Value -log(M)Mechanism of ActionActivity ReferencePublications (PubMed IDs)
Zertifikate (CoA, COO, BSE/TSE und Analyse-Diagramm)
C of A & Other Certificates(BSE/TSE, COO):
Analytical Chart:
Chemische und physikalische Eigenschaften
LöslichkeitDMSO:200 mg/mL(853.72mM;Need ultrasonic)
Lösungsrechner
Bewertungen

Kundenbewertungen

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