(±)-J 113397 - ≥98% , CAS No.217461-40-0

CAS: 217461-40-0 Cat. No.: J287289 Summenformel: C₂₄H₃₇N₃O₂ Molekulargewicht: 399.57 PubChem CID: 90488772

GRADE & PURITY ≥98%

Synonyms

(±)-1-[(3R*,4R*)-1-(Cyclooctylmethyl)-3-(hydroxymethyl)-4-piperidinyl]-3-ethyl-1,3-dihydro-2H-benzimidazol-2-one

Storage

Protected from light,Store at -20°C,Desiccated

Shipped In

Ice chest + Ice pads

Specifications

Synonyme

(±)-1-[(3R*,4R*)-1-(Cyclooctylmethyl)-3-(hydroxymethyl)-4-piperidinyl]-3-ethyl-1,3-dihydro-2H-benzimidazol-2-one

Spezifikationen & Reinheit

≥98%

Biochemische und physiologische Mechanismen

(±) - J-113397 is an effective and selective non peptide ORL1 receptor antagonist with a Ki of 1.8 nM against human cloned ORL1. J-113397 inhibits the binding of GTP γ S stimulated by nociceptin/orphan FQ to CHO cells expressing ORL1, with an IC50 value o

Storage

Protected from light,Store at -20°C,Desiccated

Verschickt in

Ice chest + Ice pads

Dieses Produkt erfordert Kühlkettenversand. Grundversand und andere Economy-Optionen sind nicht verfügbar.

Aktionsart

ANTAGONIST

Reinheit

≥98%

Namen und Kennungen

• Kanonisches Lächeln: CCN1C4=C(C=CC=C4)N([C@@H]2CCN(CC3CCCCCCC3)C[C@H]2CO)C1=O.CCN5C8=C(C=CC=C8)N([C@H]6CCN(CC7CCCCCCC7)C[C@@H]6CO)C5=O
• InChIKey: NLSVMRCGZVSAFK-SDNSQTLOSA-N
• Isomere SMILES: CCN1C2=CC=CC=C2N(C1=O)[C@@H]3CCN(C[C@H]3CO)CC4CCCCCCC4.CCN1C2=CC=CC=C2N(C1=O)[C@H]3CCN(C[C@@H]3CO)CC4CCCCCCC4
• PubChem CID: 90488772
• Molekulargewicht: 399.57

Chemische und physikalische Eigenschaften

• Löslichkeit: Solvent:DMSO, Max Conc. mg/mL: 19.98, Max Conc. mM: 50; Solvent:ethanol, Max Conc. mg/mL: 19.98, Max Conc. mM: 50
• Empfindlichkeit: Light and Moisture sensitive

Häufig gestellte Fragen

What is the purity of this product?

This product is supplied at ≥98% purity (chemical assay). Lot-specific values are stated on the Certificate of Analysis.

How should this product be stored?

Store at ?20 °C, protected from light, desiccated. Keep the container tightly closed with desiccant — the material is moisture-sensitive.

How is this product shipped?

This product ships in an insulated container with ice pads. Unpack on arrival and transfer it to the storage condition stated above.

What are the CAS number, molecular formula and molecular weight?

The CAS Number is 217461-40-0, the molecular formula is C24H37N3O2, and the molecular weight is 399.57 g/mol. InChIKey NLSVMRCGZVSAFK-SDNSQTLOSA-N.

What documentation is provided?

Available product documentation, including Certificates of Analysis (COA), Safety Data Sheets (SDS), and specification sheets, is shown in the product document area. Document availability and access follow the current site policy.