GRADE & PURITYMoligand™?Moligand™ — Aladdin's line of ligands and bioactive small molecules. Use for receptor, pathway, and binding studies needing defined small-molecule tools.10 mM in DMSO
Moligand™, 10 mM in DMSO Moligand™ for sensitive chromatographic and analytical workflows requiring minimal baseline interference.
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Storage & shipping
Store at -80°C Ships Dry ice packs + Cold packs Check lot-specific COA for exact specifications.
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Quality documents
SDS, COA, datasheet, and spec sheet available for download. Lot-specific COA accessible via lot number lookup.
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Literature proof
Cited in 0 peer-reviewed publications across chromatography, organic synthesis, and cross-coupling reactions.
Overview
MRK-016 is a selective, orally bioavailable inverse agonist of GABA A α5 receptor , with an EC 50 of 3 nM for GABA A α5, and K i s of 0.83, 0.85, 0.77?and 1.4?nM for human?GABA A ?α1β3γ2, GABA A ?α2β3γ2, GABA A ?α3β3γ2, and GABA A ?α5β3γ2, respectively; MRK-016 also readily penetrates the CNS.
Specifications
Specifications & Purity
Moligand™, 10 mM in DMSO
Storage
Store at -80°C
Shipped In
Dry ice packs + Cold packs
This product requires cold chain shipping. Ground and other economy services are not available.
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